CAPELLI, DAVIDE
CAPELLI, DAVIDE
Istituto di Cristallografia - IC
A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor gamma Binding Properties and Biological Activities
2020 Peiretti, Franck; Montanari, Roberta; Capelli, Davide; Bonardo, Bernadette; Colson, Cecilia; Amri, Ezzoubir; Grimaldi, Marina; Balaguer, Patrick; Ito, Keiichi; Roeder Robert, G; Pochetti, Giorgio; Brunel Jean, Michel
Betulinic acid is a PPARg antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis
2017 Brusotti G; Montanari R; Capelli D; Cattaneo G; Laghezza A; Tortorella P; Loiodice F; Peiretti F; Bonardo B; Paiardini A; Calleri E; Pochetti G.
Biological Screening and Crystallographic Studies of Hydroxy gamma-Lactone Derivatives to Investigate PPARgamma Phosphorylation Inhibition
2023 Capelli, D; Cazzaniga, G; Mori, M; Laghezza, A; Loiodice, F; Quaglia, M; Negro, E; Meneghetti, F; Villa, S; Montanari, R
Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy
2020 Laghezza, Antonio; Piemontese, Luca; Brunetti, Leonardo; Caradonna, Alessia; Agamennone, Mariangela; Di Pizio, Antonella; Pochetti, Giorgio; Montanari, Roberta; Capelli, Davide; Tauro, Marilena; Loiodice, Fulvio; Tortorella, Paolo
Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity
2016 Tauro M.; Laghezza A.; Loiodice F.; Piemontese L.; Caradonna A.; Capelli D.; Montanari R.; Pochetti G.; Di Pizio A.; Agamennone M.; Campestre C.; Tortorella P.
Discovery of novel chemical series of oxa-48 beta-lactamase inhibitors by high-throughput screening
2021 Garofalo B.; Prati F.; Buonfiglio R.; Coletta I.; D'atanasio N.; Molteni A.; Carettoni D.; Wanke V.; Pochetti G.; Montanari R.; Capelli D.; Milanese C.; Di Giorgio F.P.; Ombrato R.
Electrochemical and Structural Characterization of Lanthanum-Doped Hydroxyapatite: A Promising Material for Sensing Applications
2023 Cancelliere, R; Rea, G; Micheli, L; Mantegazza, P; Bauer, Em; El Khouri, A; Tempesta, E; Altomare, A; Capelli, D; Capitelli, F
Functional Nano-Hydroxyapatite for Applications in Conservation of Stony Monuments of Cultural Heritage
2020 Capitelli Francesco ; Dida Bujar ; Della Ventura Giancarlo ; Baldassarre Francesco ; Capelli Davide ; Senesi Giorgio S. ; Mele Altin ; Siliqi Dritan
Identification of the first PPARa/g able to bind to canonical and alternate sites of PPARg and to inhibit its Cdk-5-mediated phosphorylation
2018 Laghezza A.; Piemontese L.; Cerchia C.; Montanari R.; Capelli D.; Giudici M.; Crestani M.; Tortorella P.; Peiretti F.; Pochetti G.; Lavecchia A.; Loiodice F
Insights into PPARgamma Phosphorylation and Its Inhibition Mechanism
2020 Montanari R.; Capelli D.; Yamamoto K.; Awaishima H.; Nishikata K.; Barendregt A.; Heck A.J.R.; Loiodice F.; Altieri F.; Paiardini A.; Grottesi A.; Pirone L.; Pedone E.; Peiretti F.; Brunel J.M.; Itoh T.; Pochetti G.
New 2-aryloxy-3-phenyl-propanoic acids as peroxisome proliferator-activated receptors alpha/gamma dual agonists able ti up regulate the mitochondrial carnitine shuttle system gene expression.
2013 Laghezza A; Pochetti G; Lavecchia A; Fracchiolla G; Faliti S; Piemontese L; Di Giovanni C; Iacobazzi V; Infantino V; Montanari R; Capelli D; Tortorella P; Loiodice F
Novel N-(Heterocyclylphenyl)benzensulfonamide Sharing an Unreported Binding Site with T-Cell Factor 4 at the Beta-Catenin Armadillo Repeats Domain as an Anticancer Agent
2023 Nalli, Marianna; Di Magno, Laura; Wen, Yichao; Liu, Xin; D'Ambrosio, Michele; Puxeddu, Michela; Parisi, Anastasia; Sebastiani, Jessica; Sorato, Andrea; Coluccia, Antonio; Ripa, Silvia; Di Pastena, Fiorella; Capelli, Davide; Montanari, Roberta; Masci, Domiziana; Urbani, Andrea; Naro, Chiara; Sette, Claudio; Orlando, Viviana; D'Angelo, Sara; Biagioni, Stefano; Bigogno, Chiara; Dondio, Giulio; Pastore, Arianna; Stornaiuolo, Mariano; Canettieri, Gianluca; Liu, Te; Silvestri, Romano; La Regina, Giuseppe
On the Metabolically Active Form of Metaglidasen: Improved Synthesis and Investigation of Its Peculiar Activity on Peroxisome Proliferator-Activated Receptors and Skeletal Muscles.
2015 Laghezza, A; Montanari, R; Lavecchia, A; Piemontese, L; Pochetti, G; Iacobazzi, V; Infantino, V; Capelli, D; De Bellis, M; Liantonio, A; Pierno, S; Tortorella, P; Conte Camerino, D; Loiodice, F
PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc
2021 Fani Souvalidou; Dalila Boi; Davide Capelli; Federica Polverino; Grazia Marini; Roberta Montanari; Giorgio Pochetti; Angela Tramonti; Roberto Contestabile; Daniela Trisciuoglio; Patrizia Carpinelli; Camilla Ascanelli; Catherine Lindon; Alessandro De Leo; Michele Saviano; Roberto Di Santo; Roberta Costi; Giulia Guarguaglini; Alessandro Paiardini
Resveratrol and Its Metabolites Bind to PPARs
2014 Calleri, Enrica; Pochetti, Giorgio; Dossou Katina, S S; Laghezza, Antonio; Montanari, Roberta; Capelli, Davide; Prada, Ellen; Loiodice, Fulvio; Massolini, Gabriella; Bernier, Michel; Moaddel, Ruin
Screening of saponins and sapogenins from Medicago species as potential PPAR? agonists and X-ray structure of the complex PPAR?/caulophyllogenin
2016 Montanari R.; Capelli D.; Tava A.; Galli A.; Laghezza A.; Tortorella P.; Loiodice F.; Pochetti G.
Single-Nucleotide Polymorphism of PPAR, a Protein at the Crossroads of Physiological and Pathological Processes
2017 Petrosino, Maria; Lori, Laura; Pasquo, Alessandra; Lori, Clorinda; Consalvi, Valerio; Minicozzi, Velia; Morante, Silvia; Laghezza, Antonio; Giorgi, Alessandra; Capelli, Davide; Chiaraluce, Roberta
Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode.
2016 Capelli, Davide; Cerchia, Carmen; Montanari, Roberta; Loiodice, Fulvio; Tortorella, Paolo; Laghezza, Antonio; Cervoni, Laura; Pochetti, Giorgio; Lavecchia, Antonio
Structural basis of the transactivation deficiency of the human PPAR gamma F360L mutant associated with familial partial lipodystrophy
2014 Lori, Clorinda; Pasquo, Alessandra; Montanari, Roberta; Capelli, Davide; Consalvi, Valerio; Chiaraluce, Roberta; Cervoni, Laura; Loiodice, Fulvio; Laghezza, Antonio; Aschi, Massimiliano; Giorgi, Alessandra; Pochetti, Giorgio
Structural Characterization of Low-Sr-Doped Hydroxyapatite Obtained by Solid-State Synthesis
2023 Francesco Baldassarre; Angela Altomare; Ernesto Mesto; Maria Lacalamita; Bujar Dida; Altin Mele; Elvira Maria Bauer; Massimo Puzone; Emanuela Tempesta; Davide Capelli; Dritan Siliqi; Francesco Capitelli
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor gamma Binding Properties and Biological Activities | 1-gen-2020 | Peiretti, Franck; Montanari, Roberta; Capelli, Davide; Bonardo, Bernadette; Colson, Cecilia; Amri, Ezzoubir; Grimaldi, Marina; Balaguer, Patrick; Ito, Keiichi; Roeder Robert, G; Pochetti, Giorgio; Brunel Jean, Michel | |
| Betulinic acid is a PPARg antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis | 1-gen-2017 | Brusotti G; Montanari R; Capelli D; Cattaneo G; Laghezza A; Tortorella P; Loiodice F; Peiretti F; Bonardo B; Paiardini A; Calleri E; Pochetti G. | |
| Biological Screening and Crystallographic Studies of Hydroxy gamma-Lactone Derivatives to Investigate PPARgamma Phosphorylation Inhibition | 1-gen-2023 | Capelli, D; Cazzaniga, G; Mori, M; Laghezza, A; Loiodice, F; Quaglia, M; Negro, E; Meneghetti, F; Villa, S; Montanari, R | |
| Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy | 1-gen-2020 | Laghezza, Antonio; Piemontese, Luca; Brunetti, Leonardo; Caradonna, Alessia; Agamennone, Mariangela; Di Pizio, Antonella; Pochetti, Giorgio; Montanari, Roberta; Capelli, Davide; Tauro, Marilena; Loiodice, Fulvio; Tortorella, Paolo | |
| Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity | 1-gen-2016 | Tauro M.; Laghezza A.; Loiodice F.; Piemontese L.; Caradonna A.; Capelli D.; Montanari R.; Pochetti G.; Di Pizio A.; Agamennone M.; Campestre C.; Tortorella P. | |
| Discovery of novel chemical series of oxa-48 beta-lactamase inhibitors by high-throughput screening | 1-gen-2021 | Garofalo B.; Prati F.; Buonfiglio R.; Coletta I.; D'atanasio N.; Molteni A.; Carettoni D.; Wanke V.; Pochetti G.; Montanari R.; Capelli D.; Milanese C.; Di Giorgio F.P.; Ombrato R. | |
| Electrochemical and Structural Characterization of Lanthanum-Doped Hydroxyapatite: A Promising Material for Sensing Applications | 1-gen-2023 | Cancelliere, R; Rea, G; Micheli, L; Mantegazza, P; Bauer, Em; El Khouri, A; Tempesta, E; Altomare, A; Capelli, D; Capitelli, F | |
| Functional Nano-Hydroxyapatite for Applications in Conservation of Stony Monuments of Cultural Heritage | 1-gen-2020 | Capitelli Francesco ; Dida Bujar ; Della Ventura Giancarlo ; Baldassarre Francesco ; Capelli Davide ; Senesi Giorgio S. ; Mele Altin ; Siliqi Dritan | |
| Identification of the first PPARa/g able to bind to canonical and alternate sites of PPARg and to inhibit its Cdk-5-mediated phosphorylation | 1-gen-2018 | Laghezza A.; Piemontese L.; Cerchia C.; Montanari R.; Capelli D.; Giudici M.; Crestani M.; Tortorella P.; Peiretti F.; Pochetti G.; Lavecchia A.; Loiodice F | |
| Insights into PPARgamma Phosphorylation and Its Inhibition Mechanism | 1-gen-2020 | Montanari R.; Capelli D.; Yamamoto K.; Awaishima H.; Nishikata K.; Barendregt A.; Heck A.J.R.; Loiodice F.; Altieri F.; Paiardini A.; Grottesi A.; Pirone L.; Pedone E.; Peiretti F.; Brunel J.M.; Itoh T.; Pochetti G. | |
| New 2-aryloxy-3-phenyl-propanoic acids as peroxisome proliferator-activated receptors alpha/gamma dual agonists able ti up regulate the mitochondrial carnitine shuttle system gene expression. | 1-gen-2013 | Laghezza A; Pochetti G; Lavecchia A; Fracchiolla G; Faliti S; Piemontese L; Di Giovanni C; Iacobazzi V; Infantino V; Montanari R; Capelli D; Tortorella P; Loiodice F | |
| Novel N-(Heterocyclylphenyl)benzensulfonamide Sharing an Unreported Binding Site with T-Cell Factor 4 at the Beta-Catenin Armadillo Repeats Domain as an Anticancer Agent | 1-gen-2023 | Nalli, Marianna; Di Magno, Laura; Wen, Yichao; Liu, Xin; D'Ambrosio, Michele; Puxeddu, Michela; Parisi, Anastasia; Sebastiani, Jessica; Sorato, Andrea; Coluccia, Antonio; Ripa, Silvia; Di Pastena, Fiorella; Capelli, Davide; Montanari, Roberta; Masci, Domiziana; Urbani, Andrea; Naro, Chiara; Sette, Claudio; Orlando, Viviana; D'Angelo, Sara; Biagioni, Stefano; Bigogno, Chiara; Dondio, Giulio; Pastore, Arianna; Stornaiuolo, Mariano; Canettieri, Gianluca; Liu, Te; Silvestri, Romano; La Regina, Giuseppe | |
| On the Metabolically Active Form of Metaglidasen: Improved Synthesis and Investigation of Its Peculiar Activity on Peroxisome Proliferator-Activated Receptors and Skeletal Muscles. | 1-gen-2015 | Laghezza, A; Montanari, R; Lavecchia, A; Piemontese, L; Pochetti, G; Iacobazzi, V; Infantino, V; Capelli, D; De Bellis, M; Liantonio, A; Pierno, S; Tortorella, P; Conte Camerino, D; Loiodice, F | |
| PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc | 1-gen-2021 | Fani Souvalidou; Dalila Boi; Davide Capelli; Federica Polverino; Grazia Marini; Roberta Montanari; Giorgio Pochetti; Angela Tramonti; Roberto Contestabile; Daniela Trisciuoglio; Patrizia Carpinelli; Camilla Ascanelli; Catherine Lindon; Alessandro De Leo; Michele Saviano; Roberto Di Santo; Roberta Costi; Giulia Guarguaglini; Alessandro Paiardini | |
| Resveratrol and Its Metabolites Bind to PPARs | 1-gen-2014 | Calleri, Enrica; Pochetti, Giorgio; Dossou Katina, S S; Laghezza, Antonio; Montanari, Roberta; Capelli, Davide; Prada, Ellen; Loiodice, Fulvio; Massolini, Gabriella; Bernier, Michel; Moaddel, Ruin | |
| Screening of saponins and sapogenins from Medicago species as potential PPAR? agonists and X-ray structure of the complex PPAR?/caulophyllogenin | 1-gen-2016 | Montanari R.; Capelli D.; Tava A.; Galli A.; Laghezza A.; Tortorella P.; Loiodice F.; Pochetti G. | |
| Single-Nucleotide Polymorphism of PPAR, a Protein at the Crossroads of Physiological and Pathological Processes | 1-gen-2017 | Petrosino, Maria; Lori, Laura; Pasquo, Alessandra; Lori, Clorinda; Consalvi, Valerio; Minicozzi, Velia; Morante, Silvia; Laghezza, Antonio; Giorgi, Alessandra; Capelli, Davide; Chiaraluce, Roberta | |
| Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode. | 1-gen-2016 | Capelli, Davide; Cerchia, Carmen; Montanari, Roberta; Loiodice, Fulvio; Tortorella, Paolo; Laghezza, Antonio; Cervoni, Laura; Pochetti, Giorgio; Lavecchia, Antonio | |
| Structural basis of the transactivation deficiency of the human PPAR gamma F360L mutant associated with familial partial lipodystrophy | 1-gen-2014 | Lori, Clorinda; Pasquo, Alessandra; Montanari, Roberta; Capelli, Davide; Consalvi, Valerio; Chiaraluce, Roberta; Cervoni, Laura; Loiodice, Fulvio; Laghezza, Antonio; Aschi, Massimiliano; Giorgi, Alessandra; Pochetti, Giorgio | |
| Structural Characterization of Low-Sr-Doped Hydroxyapatite Obtained by Solid-State Synthesis | 1-gen-2023 | Francesco Baldassarre; Angela Altomare; Ernesto Mesto; Maria Lacalamita; Bujar Dida; Altin Mele; Elvira Maria Bauer; Massimo Puzone; Emanuela Tempesta; Davide Capelli; Dritan Siliqi; Francesco Capitelli |