MOCCIA, MARIALUISA
MOCCIA, MARIALUISA
Istituto di Endocrinologia e Oncologia Sperimentale ''G. Salvatore'' - IEOS
D898_E901 RET Deletion Is Oncogenic, Responds to Selpercatinib, and Treatment Resistance Can Arise Via RET-Independent Mechanisms
2023 Porcelli, Tommaso; Moccia, Marialuisa; De Stefano, Maria Angela; Ambrosio, Raffaele; Capoluongo, Ettore; Santoro, Massimo; Hadoux, Julien; Schlumberger, Martin; Carlomagno, Francesca; Salvatore, Domenico
Discovery of N-Trisubstituted Pyrimidine Derivatives as Type I RET and RET Gatekeeper Mutant Inhibitors with a Novel Kinase Binding Pose
2022 Zhang, Lingtian; Moccia, Marialuisa; Briggs, David C.; Bharate, Jaideep B.; Lakkaniga, Naga Rajiv; Knowles, Phillip; Yan, Wei; Tran, Phuc; Kharbanda, Anupreet; Wang, Xiuqi; Leung, Yuet-Kin; Frett, Brendan; Santoro, Massimo; Mcdonald, Neil Q.; Carlomagno, Francesca; Li, Hong-yu
Discovery of pyrazolo-thieno[3,2-d]pyrimidinylamino-phenyl acetamides as type-II pan-tropomyosin receptor kinase (TRK) inhibitors: Design, synthesis, and biological evaluation
2021 Yan, Wei; Zhang, Lingtian; Lv, Fengping; Moccia, Marialuisa; Carlomagno, Francesca; Landry, Christophe; Santoro, Massimo; Gosselet, Fabien; Frett, Brendan; Li, Hong-yu
Targeted activity of the small molecule kinase inhibitor Pz-1 towards RET and TRK kinases
2021 Moccia, Marialuisa; Yang, Donglin; Lakkaniga, Naga Rajiv; Frett, Brendan; Mcconnell, Nicholas; Zhang, Lingtian; Brescia, Annalisa; Federico, Giorgia; Zhang, Lingzhi; Salerno, Paolo; Santoro, Massimo; Li, Hong-yu; Carlomagno, Francesca
Titolo | Data di pubblicazione | Autore(i) | File |
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D898_E901 RET Deletion Is Oncogenic, Responds to Selpercatinib, and Treatment Resistance Can Arise Via RET-Independent Mechanisms | 1-gen-2023 | Porcelli, Tommaso; Moccia, Marialuisa; De Stefano, Maria Angela; Ambrosio, Raffaele; Capoluongo, Ettore; Santoro, Massimo; Hadoux, Julien; Schlumberger, Martin; Carlomagno, Francesca; Salvatore, Domenico | |
Discovery of N-Trisubstituted Pyrimidine Derivatives as Type I RET and RET Gatekeeper Mutant Inhibitors with a Novel Kinase Binding Pose | 1-gen-2022 | Zhang, Lingtian; Moccia, Marialuisa; Briggs, David C.; Bharate, Jaideep B.; Lakkaniga, Naga Rajiv; Knowles, Phillip; Yan, Wei; Tran, Phuc; Kharbanda, Anupreet; Wang, Xiuqi; Leung, Yuet-Kin; Frett, Brendan; Santoro, Massimo; Mcdonald, Neil Q.; Carlomagno, Francesca; Li, Hong-yu | |
Discovery of pyrazolo-thieno[3,2-d]pyrimidinylamino-phenyl acetamides as type-II pan-tropomyosin receptor kinase (TRK) inhibitors: Design, synthesis, and biological evaluation | 1-gen-2021 | Yan, Wei; Zhang, Lingtian; Lv, Fengping; Moccia, Marialuisa; Carlomagno, Francesca; Landry, Christophe; Santoro, Massimo; Gosselet, Fabien; Frett, Brendan; Li, Hong-yu | |
Targeted activity of the small molecule kinase inhibitor Pz-1 towards RET and TRK kinases | 1-gen-2021 | Moccia, Marialuisa; Yang, Donglin; Lakkaniga, Naga Rajiv; Frett, Brendan; Mcconnell, Nicholas; Zhang, Lingtian; Brescia, Annalisa; Federico, Giorgia; Zhang, Lingzhi; Salerno, Paolo; Santoro, Massimo; Li, Hong-yu; Carlomagno, Francesca |