MILARDI, DANILO
MILARDI, DANILO
Istituto di Cristallografia - IC - Sede Secondaria Catania
SUMO-2 activity is inhibited by non-covalent interactions with the Aβ peptide: an exploration of potential pathogenic mechanisms in Alzheimer's disease
2025 Ciaffaglione, V.; Grasso, G.; Lanza, V.; Sciacca, M. F. M.; Zimbone, S.; Giuffrida, M. L.; Iacobucci, C.; Di Ianni, A.; Calcagno, D.; Grasso, G.; Alloni, A.; Orsini, F.; Fraser, P.; Fioriti, L.; Milardi, D.
Synthesis of Ethylphosphonate Curcumin Mimics: Substituents Allow Switching Between Cytotoxic and Cytoprotective Activities
2025 Romanucci, Valeria; Pagano, Rita; Koeberle, Solveigh; Koeberle, Andreas; Bui Hoang, Minh; Di Gaetano, Sonia; Capasso, Domenica; Sciacca, Michele Francesco Maria; Lanza, Valeria; Tempra, Carmelo; Lolicato, Fabio; Zarrelli, Armando; Milardi, Danilo; Di Fabio, Giovanni
Tetra-anionic porphyrin mimics protein-protein interactions between regulatory particles and the catalytic core, allosterically activating human 20S proteasome
2025 Santoro, A. M.; Persico, M.; D'Urso, A.; Cunsolo, A.; Tkachuk, O.; Milardi, D.; Purrello, R.; Tundo, G. R.; Sbardella, D.; Osmulski, P. A.; Gaczynska, M.; Coletta, M.; Fattorusso, C.
Unveiling the Potential of a New β‐Cyclodextrin‐Suxibuzone Conjugate in Proteasome Regulation
2025 Bognanni, Noemi; Zimbone, Stefania; Giuffrida, Maria Laura; Di Natale, Giuseppe; Milardi, Danilo; Vecchio, Graziella; Lanza, Valeria
A VEGF fragment encompassing residues 10-30 inhibits A1-42 amyloid aggregation and exhibits neuroprotective properties matching the full-length protein
2024 Zimbone, Stefania; Laura Giuffrida, M; Sciacca, MICHELE FRANCESCO MARIA; Carrotta, Rita; Librizzi, Fabio; Milardi, Danilo; Grasso, Giulia
Editorial
2024 Abedini, Andisheh; Khemtemourian, Lucie; Ivanova, Magdalena; Milardi, Danilo; La Rosa, Carmelo
Exploring the therapeutic potential of Aloin: unraveling neuroprotective and anticancer mechanisms, and strategies for enhanced stability and delivery
2024 Zimbone, Stefania; Romanucci, Valeria; Zarrelli, Armando; Giuffrida, Maria Laura; Sciacca, Michele Francesco Maria.; Lanza, Valeria; Campagna, Tiziana; Maugeri, Ludovica; Petralia, Salvatore; Consoli, Grazia Maria Letizia; Di Fabio, Giovanni; Milardi, Danilo
Aβ8-20 Fragment as an Anti-Fibrillogenic and Neuroprotective Agent: Advancing toward Efficient Alzheimer’s Disease Treatment
2023 Zimbone, S.; Giuffrida, M. L.; Sabatino, G.; Di Natale, G.; Tosto, R.; Consoli, G. M. L.; Milardi, D.; Pappalardo, G.; Sciacca, M. F. M.
Electronic Circular Dichroism Detects Conformational Changes Associated with Proteasome Gating Confirmed Using AFM Imaging
2023 D'Urso, Alessandro; Purrello, Roberto; Cunsolo, Alessandra; Milardi, Danilo; Fattorusso, Caterina; Persico, Marco; Gaczynska, Maria; Osmulski Pawel, A; Santoro, ANNA MARIA
Fraisinib: a calixpyrrole derivative reducing A549 cell-derived NSCLC tumor in vivo acts as a ligand of the glycine-tRNA synthase, a new molecular target in oncology
2023 Ben Toumia, Iméne; Bachetti, Tiziana; Chekirghedira, Leila; Profumo, Aldo; Ponassi, Marco; Di Domizio, Alessandro; Izzotti, Alberto; Sciacca, Salvatore; Puglisi, Caterina; Forte, Stefano; Giuffrida, Raffaella; Colarossi, Cristina; Milardi, Danilo; Grasso, Giuseppe; Lanza, Valeria; Fiordoro, Stefano; Drago, Giacomo; Tkachenko, Kateryna; Cardinali, Barbara; Romano, Paolo; Iervasi, Erika; Vargas Gabriela, Coronel; Barboro, Paola; Kohnke Franz, Heinrich; Rosano, Camillo
Identification of a novel adiponectin receptor and opioid receptor dual acting agonist as a potential treatment for diabetic neuropathy
2023 Ma, Okf; Ronsisvalle, S; Basile, L; Xiang, Aw; Tomasella, C; Sipala, F; Pappalardo, M; Chan, Kh; Milardi, D; Ng, Rcl; Guccione, S
SASDSF2 - K48-linked diubiquitin
2023 Mangini, V; Grasso, G; Belviso, Bd; Sciacca, Mfm; Lanza, V; Caliandro, R; Milardi, D
SASDSG2 - K48-linked diubiquitin in the presence of zinc ion
2023 Mangini, V; Grasso, G; Belviso, Bd; Sciacca, Mfm; Lanza, V; Caliandro, R; Milardi, D
SASDSH2 - K48-linked diubiquitin in the presence of copper (II) ion
2023 Mangini, V; Grasso, G; Belviso, Bd; Sciacca, Mfm; Lanza, V; Caliandro, R; Milardi, D
Stretching the chains: the destabilizing impact of Cu2+ and Zn2+ ions on K48-linked diubiquitin
2023 Mangini, Vincenzo; Grasso, Giulia; Belviso, BENNY DANILO; Sciacca Michele, F M; Lanza, Valeria; Caliandro, Rocco; Milardi, Danilo
Targeting immunoproteasome in neurodegeneration: A glance to the future
2023 Tundo, Gr; Cascio, P; Milardi, D; Santoro, Am; Graziani, G; Lacal, Pm; Bocedi, A; Oddone, F; Parravano, M; Coletta, A; Coletta, M; Sbardella, D
Terpyridine Glycoconjugates and Their Metal Complexes: Antiproliferative Activity and Proteasome Inhibition
2023 Panebianco, Roberta; Viale, Maurizio; Loiacono, Fabrizio; Lanza, Valeria; Milardi, Danilo; Vecchio, Graziella
A? and Tau Interact with Metal Ions, Lipid Membranes and Peptide-Based Amyloid Inhibitors: Are These Common Features Relevant in Alzheimer's Disease?
2022 DI NATALE, Giuseppe; Sabatino, Giuseppina; Sciacca, MICHELE FRANCESCO MARIA; Tosto, Rita; Milardi, Danilo; Pappalardo, Giuseppe
beta and gamma-Cyclodextrin dimers: design, characterization and in silico studies to explore the cooperative effect of the cavities
2022 La Piana, Luana; Basile, Livia; Ragusa, Chiara; Milardi, Danilo; Zito, Valeria M. V.; Vecchio, Graziella
Corrigendum to "Silybins are stereospecific regulators of the 20S proteasome" [Bioorgan. Med. Chem. 66 (2022) 116813] (Bioorganic & Medicinal Chemistry (2022) 66, (S096808962200205X), (10.1016/j.bmc.2022.116813))
2022 Persico, Marco; Garcíaviñuales, Sara; Santoro, ANNA MARIA; Lanza, Valeria; Tundo Grazia, Raffaella; Sbardella, Diego; Coletta, Massimiliano; Romanucci, Valeria; Zarrelli, Armando; Di Fabio, Giovanni; Fattorusso, Caterina; Milardi, Danilo
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| SUMO-2 activity is inhibited by non-covalent interactions with the Aβ peptide: an exploration of potential pathogenic mechanisms in Alzheimer's disease | 1-gen-2025 | Ciaffaglione, V.; Grasso, G.; Lanza, V.; Sciacca, M. F. M.; Zimbone, S.; Giuffrida, M. L.; Iacobucci, C.; Di Ianni, A.; Calcagno, D.; Grasso, G.; Alloni, A.; Orsini, F.; Fraser, P.; Fioriti, L.; Milardi, D. | |
| Synthesis of Ethylphosphonate Curcumin Mimics: Substituents Allow Switching Between Cytotoxic and Cytoprotective Activities | 1-gen-2025 | Romanucci, Valeria; Pagano, Rita; Koeberle, Solveigh; Koeberle, Andreas; Bui Hoang, Minh; Di Gaetano, Sonia; Capasso, Domenica; Sciacca, Michele Francesco Maria; Lanza, Valeria; Tempra, Carmelo; Lolicato, Fabio; Zarrelli, Armando; Milardi, Danilo; Di Fabio, Giovanni | |
| Tetra-anionic porphyrin mimics protein-protein interactions between regulatory particles and the catalytic core, allosterically activating human 20S proteasome | 1-gen-2025 | Santoro, A. M.; Persico, M.; D'Urso, A.; Cunsolo, A.; Tkachuk, O.; Milardi, D.; Purrello, R.; Tundo, G. R.; Sbardella, D.; Osmulski, P. A.; Gaczynska, M.; Coletta, M.; Fattorusso, C. | |
| Unveiling the Potential of a New β‐Cyclodextrin‐Suxibuzone Conjugate in Proteasome Regulation | 1-gen-2025 | Bognanni, Noemi; Zimbone, Stefania; Giuffrida, Maria Laura; Di Natale, Giuseppe; Milardi, Danilo; Vecchio, Graziella; Lanza, Valeria | |
| A VEGF fragment encompassing residues 10-30 inhibits A1-42 amyloid aggregation and exhibits neuroprotective properties matching the full-length protein | 1-gen-2024 | Zimbone, Stefania; Laura Giuffrida, M; Sciacca, MICHELE FRANCESCO MARIA; Carrotta, Rita; Librizzi, Fabio; Milardi, Danilo; Grasso, Giulia | |
| Editorial | 1-gen-2024 | Abedini, Andisheh; Khemtemourian, Lucie; Ivanova, Magdalena; Milardi, Danilo; La Rosa, Carmelo | |
| Exploring the therapeutic potential of Aloin: unraveling neuroprotective and anticancer mechanisms, and strategies for enhanced stability and delivery | 1-gen-2024 | Zimbone, Stefania; Romanucci, Valeria; Zarrelli, Armando; Giuffrida, Maria Laura; Sciacca, Michele Francesco Maria.; Lanza, Valeria; Campagna, Tiziana; Maugeri, Ludovica; Petralia, Salvatore; Consoli, Grazia Maria Letizia; Di Fabio, Giovanni; Milardi, Danilo | |
| Aβ8-20 Fragment as an Anti-Fibrillogenic and Neuroprotective Agent: Advancing toward Efficient Alzheimer’s Disease Treatment | 1-gen-2023 | Zimbone, S.; Giuffrida, M. L.; Sabatino, G.; Di Natale, G.; Tosto, R.; Consoli, G. M. L.; Milardi, D.; Pappalardo, G.; Sciacca, M. F. M. | |
| Electronic Circular Dichroism Detects Conformational Changes Associated with Proteasome Gating Confirmed Using AFM Imaging | 1-gen-2023 | D'Urso, Alessandro; Purrello, Roberto; Cunsolo, Alessandra; Milardi, Danilo; Fattorusso, Caterina; Persico, Marco; Gaczynska, Maria; Osmulski Pawel, A; Santoro, ANNA MARIA | |
| Fraisinib: a calixpyrrole derivative reducing A549 cell-derived NSCLC tumor in vivo acts as a ligand of the glycine-tRNA synthase, a new molecular target in oncology | 1-gen-2023 | Ben Toumia, Iméne; Bachetti, Tiziana; Chekirghedira, Leila; Profumo, Aldo; Ponassi, Marco; Di Domizio, Alessandro; Izzotti, Alberto; Sciacca, Salvatore; Puglisi, Caterina; Forte, Stefano; Giuffrida, Raffaella; Colarossi, Cristina; Milardi, Danilo; Grasso, Giuseppe; Lanza, Valeria; Fiordoro, Stefano; Drago, Giacomo; Tkachenko, Kateryna; Cardinali, Barbara; Romano, Paolo; Iervasi, Erika; Vargas Gabriela, Coronel; Barboro, Paola; Kohnke Franz, Heinrich; Rosano, Camillo | |
| Identification of a novel adiponectin receptor and opioid receptor dual acting agonist as a potential treatment for diabetic neuropathy | 1-gen-2023 | Ma, Okf; Ronsisvalle, S; Basile, L; Xiang, Aw; Tomasella, C; Sipala, F; Pappalardo, M; Chan, Kh; Milardi, D; Ng, Rcl; Guccione, S | |
| SASDSF2 - K48-linked diubiquitin | 1-gen-2023 | Mangini, V; Grasso, G; Belviso, Bd; Sciacca, Mfm; Lanza, V; Caliandro, R; Milardi, D | |
| SASDSG2 - K48-linked diubiquitin in the presence of zinc ion | 1-gen-2023 | Mangini, V; Grasso, G; Belviso, Bd; Sciacca, Mfm; Lanza, V; Caliandro, R; Milardi, D | |
| SASDSH2 - K48-linked diubiquitin in the presence of copper (II) ion | 1-gen-2023 | Mangini, V; Grasso, G; Belviso, Bd; Sciacca, Mfm; Lanza, V; Caliandro, R; Milardi, D | |
| Stretching the chains: the destabilizing impact of Cu2+ and Zn2+ ions on K48-linked diubiquitin | 1-gen-2023 | Mangini, Vincenzo; Grasso, Giulia; Belviso, BENNY DANILO; Sciacca Michele, F M; Lanza, Valeria; Caliandro, Rocco; Milardi, Danilo | |
| Targeting immunoproteasome in neurodegeneration: A glance to the future | 1-gen-2023 | Tundo, Gr; Cascio, P; Milardi, D; Santoro, Am; Graziani, G; Lacal, Pm; Bocedi, A; Oddone, F; Parravano, M; Coletta, A; Coletta, M; Sbardella, D | |
| Terpyridine Glycoconjugates and Their Metal Complexes: Antiproliferative Activity and Proteasome Inhibition | 1-gen-2023 | Panebianco, Roberta; Viale, Maurizio; Loiacono, Fabrizio; Lanza, Valeria; Milardi, Danilo; Vecchio, Graziella | |
| A? and Tau Interact with Metal Ions, Lipid Membranes and Peptide-Based Amyloid Inhibitors: Are These Common Features Relevant in Alzheimer's Disease? | 1-gen-2022 | DI NATALE, Giuseppe; Sabatino, Giuseppina; Sciacca, MICHELE FRANCESCO MARIA; Tosto, Rita; Milardi, Danilo; Pappalardo, Giuseppe | |
| beta and gamma-Cyclodextrin dimers: design, characterization and in silico studies to explore the cooperative effect of the cavities | 1-gen-2022 | La Piana, Luana; Basile, Livia; Ragusa, Chiara; Milardi, Danilo; Zito, Valeria M. V.; Vecchio, Graziella | |
| Corrigendum to "Silybins are stereospecific regulators of the 20S proteasome" [Bioorgan. Med. Chem. 66 (2022) 116813] (Bioorganic & Medicinal Chemistry (2022) 66, (S096808962200205X), (10.1016/j.bmc.2022.116813)) | 1-gen-2022 | Persico, Marco; Garcíaviñuales, Sara; Santoro, ANNA MARIA; Lanza, Valeria; Tundo Grazia, Raffaella; Sbardella, Diego; Coletta, Massimiliano; Romanucci, Valeria; Zarrelli, Armando; Di Fabio, Giovanni; Fattorusso, Caterina; Milardi, Danilo |