BATTAGLIA, ARTURO
BATTAGLIA, ARTURO
Istituto per la Sintesi Organica e la Fotoreattivita' - ISOF
Semisynthesis, Biological Activity, and Molecular Modeling Studies of C-Ring-Modified Camptothecins
2009 Varchi, G; Samori, C; Guerrini, A; Fontana, G; Bombardelli, E; Tinelli, S; Beretta, Gl; Basili, S; Moro, S; Zunino, F; Battaglia, A
OPEN LACTONE CAMPTOTHECIN-POLYAMINE CONJUGATES
2008 Sotgiu Giovanna ; Samorì Cristian ; Guerrini Andrea ; Varchi Greta ; Beretta Giovanni Luca ; Fontana Gabriele ; Bombardelli Ezio ; Carenini Nives ; Zunino Franco ; Battaglia Arturo
Processes for the preparation of camptothecin derivatives with antitumor activity
2008 Fontana, Gabriele; Bombardelli, Ezio; Manzotti, Carla; Battaglia, Arturo; Samori, Cristian
Processes for the preparation of camptothecin derivatives with antitumor activity
2008 Fontana, Gabriele; Bombardelli, Ezio; Manzotti, Carlo; Battaglia, Arturo; Samori, Cristian
Processes for the preparation of camptothecin derivatives with antitumor activity
2008 Fontana, Gabriele; Bombardelli, Ezio; Manzotti, Carla; Battaglia, Arturo; Samori, Cristian
Synthesis of alpha(2,2),beta(3)-Diamino Acids by Double Stereodifferentiation Aldol Addition of Oxazolidinone Enolates to N-(tert-Butylsulfinyl) Imines
2008 Guerrini, Andrea; Varchi, Greta; Samorì, Cristian; Battaglia, Arturo
The Role of Polyamine Architecture on the Pharmacological Activity of Open Lactone Camptothecin-Polyamine Conjugates
2008 Samorì, Cristian; Guerrini, Andrea; Varchi, Greta; Luca Beretta, Giovanni; Fontana, Gabriele; Bombardelli, Ezio; Carenini, Nives; Zunino, Franco; Bertucci, Carlo; Fiori, Jessica; Battaglia, Arturo
Thiocamptothecin
2008 Cristian Samorì ; Andrea Guerrini ; Greta Varchi ; Franco Zunino ; Giovanni Luca Beretta ; Cristina Femoni ; Ezio Bombardelli ; Gabriele Fontana ; Arturo Battaglia
THIOCAMPTOTHECIN
2008 Varchi Greta ; Battaglia Arturo ; Samorì Cristian ; Guerrini Andrea ; Fontana Gabriele ; Bombardelli Ezio ; Zunino Franco ; Beretta Giovanni Luca
Semi-synthesis and biological activity of camptothecin tripartate conjugates
2007 Samori, Cristian; Battaglia, Arturo; Guerrini, Andrea; Varchi, Greta; Beretta Giovanni, Luca; Zunino, Franco; Fontana, Gabriele; Bombardelli, Ezio
Semi-synthesis and biological activity studies of 16a-thio-camptothecins
2007 Fontana Gabriele ; Samori Cristian ; Battaglia Arturo ; Varchi Greta ; Beretta Giovanni Luca ; Zunino Franco ; Bifulco Giuseppe ; Bombardelli Ezio
Semi-synthesis and biological activity studies of C-ring modified camptothecins and 16a-thio-camptothecins
2007 Varchi, Greta; Battaglia, Arturo; Samori, Cristian; Guerrini, Andrea; Beretta Giovanni, Luca; Zunino, Franco; Fontana, Gabriele; Bombardelli, Ezio
Synthesis of chiral beta(2,2,3)-3-amino-2-hydroxyalkanoates and 3-alkyl-3-hydroxy-beta-lactams by double asymmetric induction
2007 Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A
The first synthesis of N,O-protected b 2,2,3,3-isoserines bearing two adjacent quaternary stereogenic centers and their corresponding b -lactams
2007 Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A
Biological properties of IDN5174, a new synthetic camptothecin with the open lactone ring
2006 Beretta, Gl; Petrangolini, G; De Cesare, M; Pratesi, G; Perego, P; Tinelli, S; Tortoreto, M; Zucchetti, M; Frapolli, R; Bello, E; Manzotti, C; Fontana, G; Bombardelli, E; Battaglia, A; Samori, C; Zunino, F
Methyl taxanes: synthesis and NMR configurational assignment
2006 Battaglia, A; Dambruosop, ; C, Bassarello; G, Bifulco; G, Appendino; G, Fontana; A GomezPaloma, Guerrini
Stereoselective One-Pot Synthesis of Constrained N,O-Orthogonally Protected C-Glycosyl Norstatines [C(1')-Aminoglycosyl-1,3-dioxolan-4-ones].
2006 Guerrini, A.; Varchi, G.; Battaglia, A.
Synthesis of 7- and 10-spermine conjugates of paclitaxel and 10-deacetyl-paclitaxel as potential prodrugs
2006 Battaglia, A; Guerrini, A; Baldelli, E; Fontana, G; Varchi, G; Samori, C; Bombardelli, E
2 '-Methyl taxanes: Synthesis and NMR configurational
2005 Dambruoso, P.; Bassarello, C.; Bifulco, G.; Appendino, G.; Battaglia, A.; Guerrini, A.; Fontana, G.; GomezPaloma, L.
2?-Methyl taxanes: Synthesis and NMR configurational assignment
2005 Dambruoso Paolo, Rosario; Bassarello, Carla; Bifulco, Giuseppe; Appendino Giovanni, B; Battaglia, Arturo; Guerrini, Andrea; Fontana, Gabriele; Gomezpaloma, Luigi
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Semisynthesis, Biological Activity, and Molecular Modeling Studies of C-Ring-Modified Camptothecins | 1-gen-2009 | Varchi, G; Samori, C; Guerrini, A; Fontana, G; Bombardelli, E; Tinelli, S; Beretta, Gl; Basili, S; Moro, S; Zunino, F; Battaglia, A | |
OPEN LACTONE CAMPTOTHECIN-POLYAMINE CONJUGATES | 1-gen-2008 | Sotgiu Giovanna ; Samorì Cristian ; Guerrini Andrea ; Varchi Greta ; Beretta Giovanni Luca ; Fontana Gabriele ; Bombardelli Ezio ; Carenini Nives ; Zunino Franco ; Battaglia Arturo | |
Processes for the preparation of camptothecin derivatives with antitumor activity | 1-gen-2008 | Fontana, Gabriele; Bombardelli, Ezio; Manzotti, Carla; Battaglia, Arturo; Samori, Cristian | |
Processes for the preparation of camptothecin derivatives with antitumor activity | 1-gen-2008 | Fontana, Gabriele; Bombardelli, Ezio; Manzotti, Carlo; Battaglia, Arturo; Samori, Cristian | |
Processes for the preparation of camptothecin derivatives with antitumor activity | 1-gen-2008 | Fontana, Gabriele; Bombardelli, Ezio; Manzotti, Carla; Battaglia, Arturo; Samori, Cristian | |
Synthesis of alpha(2,2),beta(3)-Diamino Acids by Double Stereodifferentiation Aldol Addition of Oxazolidinone Enolates to N-(tert-Butylsulfinyl) Imines | 1-gen-2008 | Guerrini, Andrea; Varchi, Greta; Samorì, Cristian; Battaglia, Arturo | |
The Role of Polyamine Architecture on the Pharmacological Activity of Open Lactone Camptothecin-Polyamine Conjugates | 1-gen-2008 | Samorì, Cristian; Guerrini, Andrea; Varchi, Greta; Luca Beretta, Giovanni; Fontana, Gabriele; Bombardelli, Ezio; Carenini, Nives; Zunino, Franco; Bertucci, Carlo; Fiori, Jessica; Battaglia, Arturo | |
Thiocamptothecin | 1-gen-2008 | Cristian Samorì ; Andrea Guerrini ; Greta Varchi ; Franco Zunino ; Giovanni Luca Beretta ; Cristina Femoni ; Ezio Bombardelli ; Gabriele Fontana ; Arturo Battaglia | |
THIOCAMPTOTHECIN | 1-gen-2008 | Varchi Greta ; Battaglia Arturo ; Samorì Cristian ; Guerrini Andrea ; Fontana Gabriele ; Bombardelli Ezio ; Zunino Franco ; Beretta Giovanni Luca | |
Semi-synthesis and biological activity of camptothecin tripartate conjugates | 1-gen-2007 | Samori, Cristian; Battaglia, Arturo; Guerrini, Andrea; Varchi, Greta; Beretta Giovanni, Luca; Zunino, Franco; Fontana, Gabriele; Bombardelli, Ezio | |
Semi-synthesis and biological activity studies of 16a-thio-camptothecins | 1-gen-2007 | Fontana Gabriele ; Samori Cristian ; Battaglia Arturo ; Varchi Greta ; Beretta Giovanni Luca ; Zunino Franco ; Bifulco Giuseppe ; Bombardelli Ezio | |
Semi-synthesis and biological activity studies of C-ring modified camptothecins and 16a-thio-camptothecins | 1-gen-2007 | Varchi, Greta; Battaglia, Arturo; Samori, Cristian; Guerrini, Andrea; Beretta Giovanni, Luca; Zunino, Franco; Fontana, Gabriele; Bombardelli, Ezio | |
Synthesis of chiral beta(2,2,3)-3-amino-2-hydroxyalkanoates and 3-alkyl-3-hydroxy-beta-lactams by double asymmetric induction | 1-gen-2007 | Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A | |
The first synthesis of N,O-protected b 2,2,3,3-isoserines bearing two adjacent quaternary stereogenic centers and their corresponding b -lactams | 1-gen-2007 | Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A | |
Biological properties of IDN5174, a new synthetic camptothecin with the open lactone ring | 1-gen-2006 | Beretta, Gl; Petrangolini, G; De Cesare, M; Pratesi, G; Perego, P; Tinelli, S; Tortoreto, M; Zucchetti, M; Frapolli, R; Bello, E; Manzotti, C; Fontana, G; Bombardelli, E; Battaglia, A; Samori, C; Zunino, F | |
Methyl taxanes: synthesis and NMR configurational assignment | 1-gen-2006 | Battaglia, A; Dambruosop, ; C, Bassarello; G, Bifulco; G, Appendino; G, Fontana; A GomezPaloma, Guerrini | |
Stereoselective One-Pot Synthesis of Constrained N,O-Orthogonally Protected C-Glycosyl Norstatines [C(1')-Aminoglycosyl-1,3-dioxolan-4-ones]. | 1-gen-2006 | Guerrini, A.; Varchi, G.; Battaglia, A. | |
Synthesis of 7- and 10-spermine conjugates of paclitaxel and 10-deacetyl-paclitaxel as potential prodrugs | 1-gen-2006 | Battaglia, A; Guerrini, A; Baldelli, E; Fontana, G; Varchi, G; Samori, C; Bombardelli, E | |
2 '-Methyl taxanes: Synthesis and NMR configurational | 1-gen-2005 | Dambruoso, P.; Bassarello, C.; Bifulco, G.; Appendino, G.; Battaglia, A.; Guerrini, A.; Fontana, G.; GomezPaloma, L. | |
2?-Methyl taxanes: Synthesis and NMR configurational assignment | 1-gen-2005 | Dambruoso Paolo, Rosario; Bassarello, Carla; Bifulco, Giuseppe; Appendino Giovanni, B; Battaglia, Arturo; Guerrini, Andrea; Fontana, Gabriele; Gomezpaloma, Luigi |