BATTAGLIA, ARTURO
BATTAGLIA, ARTURO
Istituto per la Sintesi Organica e la Fotoreattivita' - ISOF
Semisynthesis, Biological Activity, and Molecular Modeling Studies of C-Ring-Modified Camptothecins
2009 Varchi, G; Samori, C; Guerrini, A; Fontana, G; Bombardelli, E; Tinelli, S; Beretta, Gl; Basili, S; Moro, S; Zunino, F; Battaglia, A
Synthesis of alpha(2,2),beta(3)-Diamino Acids by Double Stereodifferentiation Aldol Addition of Oxazolidinone Enolates to N-(tert-Butylsulfinyl) Imines
2008 Guerrini, Andrea; Varchi, Greta; Samorì, Cristian; Battaglia, Arturo
The Role of Polyamine Architecture on the Pharmacological Activity of Open Lactone Camptothecin-Polyamine Conjugates
2008 Samorì, Cristian; Guerrini, Andrea; Varchi, Greta; Luca Beretta, Giovanni; Fontana, Gabriele; Bombardelli, Ezio; Carenini, Nives; Zunino, Franco; Bertucci, Carlo; Fiori, Jessica; Battaglia, Arturo
Thiocamptothecin
2008 Cristian Samorì ; Andrea Guerrini ; Greta Varchi ; Franco Zunino ; Giovanni Luca Beretta ; Cristina Femoni ; Ezio Bombardelli ; Gabriele Fontana ; Arturo Battaglia
Synthesis of chiral beta(2,2,3)-3-amino-2-hydroxyalkanoates and 3-alkyl-3-hydroxy-beta-lactams by double asymmetric induction
2007 Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A
The first synthesis of N,O-protected b 2,2,3,3-isoserines bearing two adjacent quaternary stereogenic centers and their corresponding b -lactams
2007 Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A
Biological properties of IDN5174, a new synthetic camptothecin with the open lactone ring
2006 Beretta, Gl; Petrangolini, G; De Cesare, M; Pratesi, G; Perego, P; Tinelli, S; Tortoreto, M; Zucchetti, M; Frapolli, R; Bello, E; Manzotti, C; Fontana, G; Bombardelli, E; Battaglia, A; Samori, C; Zunino, F
Methyl taxanes: synthesis and NMR configurational assignment
2006 Battaglia, A; Dambruosop, ; C, Bassarello; G, Bifulco; G, Appendino; G, Fontana; A GomezPaloma, Guerrini
Stereoselective One-Pot Synthesis of Constrained N,O-Orthogonally Protected C-Glycosyl Norstatines [C(1')-Aminoglycosyl-1,3-dioxolan-4-ones].
2006 Guerrini, A.; Varchi, G.; Battaglia, A.
Synthesis of 7- and 10-spermine conjugates of paclitaxel and 10-deacetyl-paclitaxel as potential prodrugs
2006 Battaglia, A; Guerrini, A; Baldelli, E; Fontana, G; Varchi, G; Samori, C; Bombardelli, E
2 '-Methyl taxanes: Synthesis and NMR configurational
2005 Dambruoso, P.; Bassarello, C.; Bifulco, G.; Appendino, G.; Battaglia, A.; Guerrini, A.; Fontana, G.; GomezPaloma, L.
2?-Methyl taxanes: Synthesis and NMR configurational assignment
2005 Dambruoso Paolo, Rosario; Bassarello, Carla; Bifulco, Giuseppe; Appendino Giovanni, B; Battaglia, Arturo; Guerrini, Andrea; Fontana, Gabriele; Gomezpaloma, Luigi
Advances in the universal NMR database approach. 2 '- substituted taxanes as probes for an improved protocol of diastereomeric differentiation
2005 Battaglia, A; P, Dambruoso; C, Bassarello; G, Bifulco; G, Appendino; Fontana, G; Gomezpaloma,
Selective Synthesis of 14 Beta-Amino Taxanes
2005 Battaglia A; Baldelli E; Bombardelli E; Carenzi G; Fontana G; Gelmi Ml; Guerrini A; Pocar D
Synthesis of deserpidine from reserpine
2005 Varchi, Greta; Battaglia, Arturo; Samor, Cristian; Baldelli, Eleonora; Danieli, Bruno; Fontana, Gabriele; Guerrini, Andrea; Bombardelli, Ezio
New Taxane Derivatives: Synthesis of Baccatin[14,1-d]furan-2-one Nucleus and Its Condensation with the Norstatine Side Chain
2004 Eleonora Baldelli;Arturo Battaglia;Ezio Bombardelli; Giacomo Carenzi;Gabriele Fontana; Maria Luisa Gelmi; Andrea Guerrini;Donato Pocar
Synthesis of Optically Active Constrained 2-Substituted Norstatines: A Straightforward Application of Seebach s SRS Synthetic Principle
2004 Arturo Battaglia;Andrea Guerrini;Carlo Bertucci
Diastereoselective 14 beta-hydroxylation of baccatin III derivatives
2003 Battaglia, A; Baldelli, E; Bombardelli, E; Carenzi, G; Fontana, G; Gambini, A; Gelmi, Ml; Guerrini, A; Pocar, D
Semi-synthesis of 14 beta-OH baccatin III-1,14-carbonate from 10-deacetyl baccatin III (DAB)
2003 Battaglia, A; Baldelli, E; Bombardelli, E; Carenzi, D; Gelmi, Ml; Guerrini, A; Fontana, G; Pocar, D
Synthesis and biological evaluation of 2 '-methyl taxoids derived from baccatin III and 14 beta-OH-baccatin III 1,14-carbonate
2003 Battaglia A; Bernacki RJ; Bertucci C; Bombardelli E; Cimitan S; Ferlini C; Fontana G; Guerrini A; Riva A
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Semisynthesis, Biological Activity, and Molecular Modeling Studies of C-Ring-Modified Camptothecins | 1-gen-2009 | Varchi, G; Samori, C; Guerrini, A; Fontana, G; Bombardelli, E; Tinelli, S; Beretta, Gl; Basili, S; Moro, S; Zunino, F; Battaglia, A | |
Synthesis of alpha(2,2),beta(3)-Diamino Acids by Double Stereodifferentiation Aldol Addition of Oxazolidinone Enolates to N-(tert-Butylsulfinyl) Imines | 1-gen-2008 | Guerrini, Andrea; Varchi, Greta; Samorì, Cristian; Battaglia, Arturo | |
The Role of Polyamine Architecture on the Pharmacological Activity of Open Lactone Camptothecin-Polyamine Conjugates | 1-gen-2008 | Samorì, Cristian; Guerrini, Andrea; Varchi, Greta; Luca Beretta, Giovanni; Fontana, Gabriele; Bombardelli, Ezio; Carenini, Nives; Zunino, Franco; Bertucci, Carlo; Fiori, Jessica; Battaglia, Arturo | |
Thiocamptothecin | 1-gen-2008 | Cristian Samorì ; Andrea Guerrini ; Greta Varchi ; Franco Zunino ; Giovanni Luca Beretta ; Cristina Femoni ; Ezio Bombardelli ; Gabriele Fontana ; Arturo Battaglia | |
Synthesis of chiral beta(2,2,3)-3-amino-2-hydroxyalkanoates and 3-alkyl-3-hydroxy-beta-lactams by double asymmetric induction | 1-gen-2007 | Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A | |
The first synthesis of N,O-protected b 2,2,3,3-isoserines bearing two adjacent quaternary stereogenic centers and their corresponding b -lactams | 1-gen-2007 | Guerrini, A; Varchi, G; Rizzo, D; Samori, C; Battaglia, A | |
Biological properties of IDN5174, a new synthetic camptothecin with the open lactone ring | 1-gen-2006 | Beretta, Gl; Petrangolini, G; De Cesare, M; Pratesi, G; Perego, P; Tinelli, S; Tortoreto, M; Zucchetti, M; Frapolli, R; Bello, E; Manzotti, C; Fontana, G; Bombardelli, E; Battaglia, A; Samori, C; Zunino, F | |
Methyl taxanes: synthesis and NMR configurational assignment | 1-gen-2006 | Battaglia, A; Dambruosop, ; C, Bassarello; G, Bifulco; G, Appendino; G, Fontana; A GomezPaloma, Guerrini | |
Stereoselective One-Pot Synthesis of Constrained N,O-Orthogonally Protected C-Glycosyl Norstatines [C(1')-Aminoglycosyl-1,3-dioxolan-4-ones]. | 1-gen-2006 | Guerrini, A.; Varchi, G.; Battaglia, A. | |
Synthesis of 7- and 10-spermine conjugates of paclitaxel and 10-deacetyl-paclitaxel as potential prodrugs | 1-gen-2006 | Battaglia, A; Guerrini, A; Baldelli, E; Fontana, G; Varchi, G; Samori, C; Bombardelli, E | |
2 '-Methyl taxanes: Synthesis and NMR configurational | 1-gen-2005 | Dambruoso, P.; Bassarello, C.; Bifulco, G.; Appendino, G.; Battaglia, A.; Guerrini, A.; Fontana, G.; GomezPaloma, L. | |
2?-Methyl taxanes: Synthesis and NMR configurational assignment | 1-gen-2005 | Dambruoso Paolo, Rosario; Bassarello, Carla; Bifulco, Giuseppe; Appendino Giovanni, B; Battaglia, Arturo; Guerrini, Andrea; Fontana, Gabriele; Gomezpaloma, Luigi | |
Advances in the universal NMR database approach. 2 '- substituted taxanes as probes for an improved protocol of diastereomeric differentiation | 1-gen-2005 | Battaglia, A; P, Dambruoso; C, Bassarello; G, Bifulco; G, Appendino; Fontana, G; Gomezpaloma, | |
Selective Synthesis of 14 Beta-Amino Taxanes | 1-gen-2005 | Battaglia A; Baldelli E; Bombardelli E; Carenzi G; Fontana G; Gelmi Ml; Guerrini A; Pocar D | |
Synthesis of deserpidine from reserpine | 1-gen-2005 | Varchi, Greta; Battaglia, Arturo; Samor, Cristian; Baldelli, Eleonora; Danieli, Bruno; Fontana, Gabriele; Guerrini, Andrea; Bombardelli, Ezio | |
New Taxane Derivatives: Synthesis of Baccatin[14,1-d]furan-2-one Nucleus and Its Condensation with the Norstatine Side Chain | 1-gen-2004 | Eleonora Baldelli;Arturo Battaglia;Ezio Bombardelli; Giacomo Carenzi;Gabriele Fontana; Maria Luisa Gelmi; Andrea Guerrini;Donato Pocar | |
Synthesis of Optically Active Constrained 2-Substituted Norstatines: A Straightforward Application of Seebach s SRS Synthetic Principle | 1-gen-2004 | Arturo Battaglia;Andrea Guerrini;Carlo Bertucci | |
Diastereoselective 14 beta-hydroxylation of baccatin III derivatives | 1-gen-2003 | Battaglia, A; Baldelli, E; Bombardelli, E; Carenzi, G; Fontana, G; Gambini, A; Gelmi, Ml; Guerrini, A; Pocar, D | |
Semi-synthesis of 14 beta-OH baccatin III-1,14-carbonate from 10-deacetyl baccatin III (DAB) | 1-gen-2003 | Battaglia, A; Baldelli, E; Bombardelli, E; Carenzi, D; Gelmi, Ml; Guerrini, A; Fontana, G; Pocar, D | |
Synthesis and biological evaluation of 2 '-methyl taxoids derived from baccatin III and 14 beta-OH-baccatin III 1,14-carbonate | 1-gen-2003 | Battaglia A; Bernacki RJ; Bertucci C; Bombardelli E; Cimitan S; Ferlini C; Fontana G; Guerrini A; Riva A |