PESARESI, ALESSANDRO
PESARESI, ALESSANDRO
Istituto di Cristallografia - IC
Mixed and non-competitive enzyme inhibition: underlying mechanisms andmechanistic irrelevance of the formal two-site model
2023 Pesaresi, Alessandro
Nonallosteric activation of posttranslational modification enzymes by active site-directed inhibitors
2023 Pesaresi, Alessandro
Kinetic and structural studies on the inhibition of acetylcholinesterase and butyrylcholinesterase by a series of multitarget-directed galantamine-peptide derivatives
2022 Pesaresi, A; Lamba, D; Vezenkov, L; Tsekova, D; Lozanov, V
Kinetic Modeling of Time-Dependent Enzyme Inhibition by Pre-Steady-State Analysis of Progress Curves: The Case Study of the Anti-Alzheimer's Drug Galantamine
2022 Doriano Lamba ;Alessandro Pesaresi
Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease
2019 Chalupova K.; Korabecny J.; Bartolini M.; Monti B.; Lamba D.; Caliandro R.; Pesaresi A.; Brazzolotto X.; Gastellier A.J.; Nachon F.; Pejchal J.; Jarosova M.; Hepnarova V.; Jun D.; Hrabinova M.; Dolezal R.; Zdarova Karasova J.; Mzik M.; Kristofikova Z.; Misik J.; Muckova L.; Jost P.; Soukup O.; Benkova M.; Setnicka V.; Habartova L.; Chvojkova M.; Kleteckova L.; Vales K.; Mezeiova E.; Uliassi E.; Valis M.; Nepovimova E.; Bolognesi M.L.; Kuca K.
"Kinetic and structural studies on the interactions of Torpedo californica acetylcholinesterase with two donepezil-like rigid Analogues"
2018 Caliandro R.; Pesaresi A.; Cariati L. Procopio A.; Oliverio M.; Lamba D.
Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease:Design, Synthesis, Biological Evaluation and X-ray Crystallography
2016 Zha, Xiaoming; Lamba, Doriano; Zhanga, Lili; A, Yinghan Lou; D, ; Xua, Changxu; Dikanga, ; Chen, Li; Xu, Yungen; Zhang, Luyong; De Simone, Angela; B, Sarah Samez; F, ; Pesaresi, Alessandro; Stojan, Jure; G Lopez, Manuela; Egea, Javier; Vincenzaandrisano, ; Bartolini, Manuela
Multitarget Drug Design Strategy: Quinone-Tacrine Hybrids Designed To Block Amyloid-beta Aggregation and To Exert Anticholinesterase and Antioxidant Effects
2014 Nepovímová, Eugenie; Uliassi, Elisa; Korábecný, Jan; PeñaAltamira, Luis Emiliano; Samez, Sarah; Pesaresi, Alessandro; Garcia, Gregory E.; Bartolini, Manuela; Andrisano, Vincenza; Bergamini, Christian; Fato, Romana; Lamba, Doriano; Roberti, Marinella; Kuca, Kamil; Monti, Barbara; Bolognesi, M. L.
Evaluation and computational characterization of the facilitated transport of Glc carbon C-1 oxime reactivators across a blood brain barrier model
2013 Bhonsle, ; J, B; Causey, R; Oyler, ; B, L; Bartolucci, C; Lamba, D; Pesaresi, A; Bhamare, ; N, K; Soojhawon, I; Garcia, ; G, E
Role of metal ions on the activity of Mycobacterium tuberculosis pyrazinamidase
2012 Sheen P; Ferrer P; Gilman; R H; Christiansen G; MorenoRomán P; Gutiérrez; A H; Sotelo J; Evangelista W; Fuentes P; Rueda D; Flores M; Olivera P; Solis J; Pesaresi A; Lamba D; Zimic; M
Isolation, characterization, and heterologous expression of a carboxylesterase of Pseudomonas aeruginosa PAO1.
2005 Pesaresi, A; Devescovi, G; Lamba, D; Venturi, V; Degrassi, G
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Mixed and non-competitive enzyme inhibition: underlying mechanisms andmechanistic irrelevance of the formal two-site model | 1-gen-2023 | Pesaresi, Alessandro | |
| Nonallosteric activation of posttranslational modification enzymes by active site-directed inhibitors | 1-gen-2023 | Pesaresi, Alessandro | |
| Kinetic and structural studies on the inhibition of acetylcholinesterase and butyrylcholinesterase by a series of multitarget-directed galantamine-peptide derivatives | 1-gen-2022 | Pesaresi, A; Lamba, D; Vezenkov, L; Tsekova, D; Lozanov, V | |
| Kinetic Modeling of Time-Dependent Enzyme Inhibition by Pre-Steady-State Analysis of Progress Curves: The Case Study of the Anti-Alzheimer's Drug Galantamine | 1-gen-2022 | Doriano Lamba ;Alessandro Pesaresi | |
| Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease | 1-gen-2019 | Chalupova K.; Korabecny J.; Bartolini M.; Monti B.; Lamba D.; Caliandro R.; Pesaresi A.; Brazzolotto X.; Gastellier A.J.; Nachon F.; Pejchal J.; Jarosova M.; Hepnarova V.; Jun D.; Hrabinova M.; Dolezal R.; Zdarova Karasova J.; Mzik M.; Kristofikova Z.; Misik J.; Muckova L.; Jost P.; Soukup O.; Benkova M.; Setnicka V.; Habartova L.; Chvojkova M.; Kleteckova L.; Vales K.; Mezeiova E.; Uliassi E.; Valis M.; Nepovimova E.; Bolognesi M.L.; Kuca K. | |
| "Kinetic and structural studies on the interactions of Torpedo californica acetylcholinesterase with two donepezil-like rigid Analogues" | 1-gen-2018 | Caliandro R.; Pesaresi A.; Cariati L. Procopio A.; Oliverio M.; Lamba D. | |
| Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease:Design, Synthesis, Biological Evaluation and X-ray Crystallography | 1-gen-2016 | Zha, Xiaoming; Lamba, Doriano; Zhanga, Lili; A, Yinghan Lou; D, ; Xua, Changxu; Dikanga, ; Chen, Li; Xu, Yungen; Zhang, Luyong; De Simone, Angela; B, Sarah Samez; F, ; Pesaresi, Alessandro; Stojan, Jure; G Lopez, Manuela; Egea, Javier; Vincenzaandrisano, ; Bartolini, Manuela | |
| Multitarget Drug Design Strategy: Quinone-Tacrine Hybrids Designed To Block Amyloid-beta Aggregation and To Exert Anticholinesterase and Antioxidant Effects | 1-gen-2014 | Nepovímová, Eugenie; Uliassi, Elisa; Korábecný, Jan; PeñaAltamira, Luis Emiliano; Samez, Sarah; Pesaresi, Alessandro; Garcia, Gregory E.; Bartolini, Manuela; Andrisano, Vincenza; Bergamini, Christian; Fato, Romana; Lamba, Doriano; Roberti, Marinella; Kuca, Kamil; Monti, Barbara; Bolognesi, M. L. | |
| Evaluation and computational characterization of the facilitated transport of Glc carbon C-1 oxime reactivators across a blood brain barrier model | 1-gen-2013 | Bhonsle, ; J, B; Causey, R; Oyler, ; B, L; Bartolucci, C; Lamba, D; Pesaresi, A; Bhamare, ; N, K; Soojhawon, I; Garcia, ; G, E | |
| Role of metal ions on the activity of Mycobacterium tuberculosis pyrazinamidase | 1-gen-2012 | Sheen P; Ferrer P; Gilman; R H; Christiansen G; MorenoRomán P; Gutiérrez; A H; Sotelo J; Evangelista W; Fuentes P; Rueda D; Flores M; Olivera P; Solis J; Pesaresi A; Lamba D; Zimic; M | |
| Isolation, characterization, and heterologous expression of a carboxylesterase of Pseudomonas aeruginosa PAO1. | 1-gen-2005 | Pesaresi, A; Devescovi, G; Lamba, D; Venturi, V; Degrassi, G |