AUZZAS, LUCIANA
AUZZAS, LUCIANA
Istituto di Chimica Biomolecolare - ICB - Sede Pozzuoli
1) Non-Natural Macrocyclic Inhibitors of Histone Deacetylase. 2) Rationally Designed Passepartout Agents for System-Biology Diseases: Structure-, Fragment- and Function-Based Approaches towards the Rational Design of Multitarget Ligands. Proapoptotic Antiangiogenic Dual Inhibitors of Protein Kinases and XIAP. 3) Targeting RGD-Recognizing Integrins. Synthesis and Biomedical Applications of Pyrrolidine and Cyclopentane-Based RGD Integrin Binders and Conjugates.
2009 Hanessian, S; Auzzas, L; Larsson, A; Giannini, G; Pisano, C Auzzas L Larsson A; Amodeo, P; Vitale, ROSA MARIA; R Rassu, G; Auzzas, L Casiraghi G
4-Aminoproline-based arginine-glycine-aspartate integrin binders with exposed ligation points: practical in-solution synthesis, conjugation and binding affinity evaluation
2009 Battistini, Lucia; Burreddu, Paola; Carta, Paola; Rassu, GLORIA MARIA RITA; Auzzas, Luciana; Curti, Claudio; Zanardi, Franca; Manzoni, LEONARDO PIERPAOLO; Araldi Elena, M V; Scolastico, Carlo; Casiraghi, Giovanni
A New Enantioselective Entry to Cycloeptane Polyols
2005 Curti, C; Sartori, A; Zanardi, F; Battistini, L; Rassu, G; Auzzas, L; Roggio, A M; Casiraghi, G
A Short Entry to Novel (2)-Methyl Branched 4a-Carbafuranoses
2003 Rassu, G; Auzzas, L; Zambrano, V; Burreddu, P; Battistini, L; Curti, C
A short entry to novel C(2)-methyl branched 4a-carbafuranoses
2003 Rassu, Gloria; Auzzas, Luciana; Zambrano, Vincenzo; Burreddu, Paola; Battistini, Lucia; Curti, Claudio
Advances in Chemical Synthesis of Carbasugars and Analogues
2003 Rassu, G; Auzzas, L; Pinna, L; Battistini, L; Curti, C
Advances in Chemical Synthesis of Carbasugars and Analogues.
2003 Rassu, G.; Auzzas, L.; Pinna, L.; Battistini, L.; Curti, C.
Advances in the Chemical Synthesis of Medium-sized Cyclitols
2004 Rassu, G; Auzzas, L; Battistini, L; Casiraghi, ; G,
Alternative and Expedient Asymmetric Syntheses of L-(+)-noviose.
2008 Hanessian, S; Auzzas, L
Amide Compounds and Their Use as Antitumor Agents. Eur. Pat. Appl. No. 07104071
2007 Hanessian, S; Auzzas, L; Giannini, G; Vesci, L; Pisano, C
Amide Compounds and Their Use as Antitumor Agents. WO2008110583
2008 Hanessian, S; Auzzas, L; Giannini, G; Pisano, C; Vesci, L; Cabri, W
Anti-inflammatory and analgesic amides: New developments
2000 Palomba, M; Pau, A; Boatto, G; Asproni, B; Auzzas, L; Cerri, R; Arenare, L; Filippelli, W; Falcone, G; Motola, G
Antidermatophytic action of new 1-naphthylmethyl and benzo[b]thiophen-7-ylmethyl hydrazones related to inhibitors of squalene epoxidase.
2000 Auzzas, L.; Palomba, M.; Manconi, P.; Pau, A.; Becciu, A.; Cerri, R.; Tullio, V.; Roana, J.; Carlone, N.
Attività Antidermatofitica di Nuovi Benzo[b]tiofenil-7-metil Idrazoni Strutturalmente Correlati agli Antimicotici Inibitori dello squalene epoxidasi
2000 Gian Piera Linaldeddu; Riccardo Cerri; Luciana Auzzas; Gianpiero Boatto
Battling Cancer: A Fragment-Based Approach towards the Design of Multitargeted Ligands
2010 Edvinsson, S.; Larsson, A.; Auzzas, L.
Ciclopeptidi Ibridi Contenenti Amminoacidi Cicloalcanici, e Loro Preparazione ed Uso.
2005 Casiraghi, G; Rassu, G; Auzzas, L; Battistini, L; Zanardi, F; Curti, C; Nicastro, G; Belvisi, L; Castorina, M; Giannini, G; Pisano, C
Design of multitargeted ligands
2014 Andreas Larsson; Sofie Knutsson; Luciana Auzzas
Discovery of Subnanomolar Arginine-Glycine-Aspartate-Based aVb3/aVb5 Integrin Binders Embedding 4-Aminoproline Residues.
2008 Zanardi, F; Burreddu, P; Rassu, G; Auzzas, L; Battistini, L; Curti, C; Sartori, A; Nicastro, G; Menchi, G; Cini, N; Bottoncetti, A; Raspanti, S; Casiraghi, G
Enantioselective Total Synthesis of (1R,3S,4R,5R)-1-Amino-4,5-dihydroxycyclopentane-1,3-dicarboxylic Acid. A Full-Aldol Access to Carbaketose Derivatives
2004 Battistini, L; Curti, C; Zanardi, F; Rassu, G; Auzzas, L; Casiraghi, G
Exploring Alternative Zn-binding Groups in the Design of HDAC inhibitors: Squaric Acid, N-Hydroxyurea, and Oxazoline Analogues of SAHA
2006 Hanessian S.; Vinci V.; Auzzas L.; Marzi M.; Giannini G.