AUZZAS, LUCIANA
AUZZAS, LUCIANA
Istituto di Chimica Biomolecolare - ICB - Sede Secondaria Sassari
Non-Natural Macrocyclic Inhibitors of Histone Deacetylases: Design, Synthesis, and Activity
2010 Auzzas, L; Larsson, A; Matera, R; Baraldi, A; Deschênessimard, B; Giannini, G; Cabri, W; Battistuzzi, G; Gallo, G; Ciacci, A; Vesci, L; Pisano, C; Hanessian, S
Targeting alphaVbeta3 Integrin: Design and Applications of Mono- and Multifunctional RGD-Based Peptides and Semipeptides
2010 Auzzas, L; Zanardi, F; Battistini, L; Burreddu, P; Carta, P; Rassu, G; Curti, C; Casiraghi, G
Vorinostat-Like Molecules as Structural, Stereochemical, and Pharmacological Tools
2010 Hanessian, S; Auzzas, L; Larsson, A; Zhang, J; Giannini, G; Gallo, G; Ciacci, A; Cabri, W
4-Aminoproline-based arginine-glycine-aspartate integrin binders with exposed ligation points: practical in-solution synthesis, conjugation and binding affinity evaluation
2009 Battistini, Lucia; Burreddu, Paola; Carta, Paola; Rassu, GLORIA MARIA RITA; Auzzas, Luciana; Curti, Claudio; Zanardi, Franca; Manzoni, LEONARDO PIERPAOLO; Araldi Elena, M V; Scolastico, Carlo; Casiraghi, Giovanni
Alternative and Expedient Asymmetric Syntheses of L-(+)-noviose.
2008 Hanessian, S; Auzzas, L
Discovery of Subnanomolar Arginine-Glycine-Aspartate-Based aVb3/aVb5 Integrin Binders Embedding 4-Aminoproline Residues.
2008 Zanardi, F; Burreddu, P; Rassu, G; Auzzas, L; Battistini, L; Curti, C; Sartori, A; Nicastro, G; Menchi, G; Cini, N; Bottoncetti, A; Raspanti, S; Casiraghi, G
The Practice of Ring Constraint in Peptidomimetics Using Bicyclic and Polycyclic Amino Acids.
2008 Hanessian, S; Auzzas, L
omega-Alkoxy analogues of SAHA(vorinostat) as inhibitors of HDAC: a study of chain-lenght and stereochemical dependence.
2007 Hanessian S.; Auzzas L.; Giannini G.; Marzi M.; Cabri W.; Barbarino M.; Vesci L.; Pisano C.
Exploring Alternative Zn-binding Groups in the Design of HDAC inhibitors: Squaric Acid, N-Hydroxyurea, and Oxazoline Analogues of SAHA
2006 Hanessian S.; Vinci V.; Auzzas L.; Marzi M.; Giannini G.
New Enantioselective Entry to Cycloheptane Amino Acid Polyols.
2006 Curti C.; Zanardi F.; Battistini L.; Sartori A.; Rassu G.; Auzzas L.; Roggio A.; Pinna L.; Casiraghi G.
Grafting Aminocyclopentane Carboxylic Acids onto the RGD Tripeptide Sequence Generates Low Nanomolar aVb3/aVb5 Integrin Dual Binders.
2005 Casiraghi, G; Rassu, G; Auzzas, L; Burreddu, P; Gaetani, E; Battistini, L; Zanardi, F; Curti, C; Nicastro, G; Belvisi, L; Motto, I; Castorina, M; Giannini, G; Pisano, C
Advances in the Chemical Synthesis of Medium-sized Cyclitols
2004 Rassu, G; Auzzas, L; Battistini, L; Casiraghi, ; G,
Enantioselective Total Synthesis of (1R,3S,4R,5R)-1-Amino-4,5-dihydroxycyclopentane-1,3-dicarboxylic Acid. A Full-Aldol Access to Carbaketose Derivatives
2004 Battistini, L; Curti, C; Zanardi, F; Rassu, G; Auzzas, L; Casiraghi, G
Variable Strategy toward Carbasugars and Relatives. 6. Diastereoselective Synthesis of 2-Deoxy-2-amino-5a-carba-beta-L-mannopyranuronic Acid and 2-Deoxy-2-amino-5a-carba-beta-L-mannopyranose
2004 Rassu G.; Auzzas L.; Zambrano V.; Burreddu P.; Pinna L.; Battistini L.; Zanardi F.; Casiraghi G.
A Short Entry to Novel (2)-Methyl Branched 4a-Carbafuranoses
2003 Rassu, G; Auzzas, L; Zambrano, V; Burreddu, P; Battistini, L; Curti, C
A short entry to novel C(2)-methyl branched 4a-carbafuranoses
2003 Rassu, Gloria; Auzzas, Luciana; Zambrano, Vincenzo; Burreddu, Paola; Battistini, Lucia; Curti, Claudio
Advances in Chemical Synthesis of Carbasugars and Analogues
2003 Rassu, G; Auzzas, L; Pinna, L; Battistini, L; Curti, C
Isopavines as a New Class of Morphinomimetics
2003 Casiraghi, G; Zanardi, F; Auzzas, L; Appendino, G
Variable Strategy toward Carbasugars and Relatives. 5. Focus on Preparation of Chiral Nonracemic Medium-Sized Carbocycles
2003 Rassu, Gloria; Auzzas, Luciana; Pinna, Luigi; Zambrano, Vincenzo; Zanardi, Franca; Battistini, Lucia; Gaetani, Enrico; Curti, Claudio; Casiraghi, Giovanni
Variable Strategy towards Carbasugars and Relatives. 5. Focus on Preparation of Chiral Nonracemic Medium-Sized Carbocycles
2003 Rassu, G; Auzzas, L; Pinna, L; Zambrano, V; Zanardi, F; Battistini, L; Gaetani, E; Curti, C; Casiraghi, G
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Non-Natural Macrocyclic Inhibitors of Histone Deacetylases: Design, Synthesis, and Activity | 1-gen-2010 | Auzzas, L; Larsson, A; Matera, R; Baraldi, A; Deschênessimard, B; Giannini, G; Cabri, W; Battistuzzi, G; Gallo, G; Ciacci, A; Vesci, L; Pisano, C; Hanessian, S | |
| Targeting alphaVbeta3 Integrin: Design and Applications of Mono- and Multifunctional RGD-Based Peptides and Semipeptides | 1-gen-2010 | Auzzas, L; Zanardi, F; Battistini, L; Burreddu, P; Carta, P; Rassu, G; Curti, C; Casiraghi, G | |
| Vorinostat-Like Molecules as Structural, Stereochemical, and Pharmacological Tools | 1-gen-2010 | Hanessian, S; Auzzas, L; Larsson, A; Zhang, J; Giannini, G; Gallo, G; Ciacci, A; Cabri, W | |
| 4-Aminoproline-based arginine-glycine-aspartate integrin binders with exposed ligation points: practical in-solution synthesis, conjugation and binding affinity evaluation | 1-gen-2009 | Battistini, Lucia; Burreddu, Paola; Carta, Paola; Rassu, GLORIA MARIA RITA; Auzzas, Luciana; Curti, Claudio; Zanardi, Franca; Manzoni, LEONARDO PIERPAOLO; Araldi Elena, M V; Scolastico, Carlo; Casiraghi, Giovanni | |
| Alternative and Expedient Asymmetric Syntheses of L-(+)-noviose. | 1-gen-2008 | Hanessian, S; Auzzas, L | |
| Discovery of Subnanomolar Arginine-Glycine-Aspartate-Based aVb3/aVb5 Integrin Binders Embedding 4-Aminoproline Residues. | 1-gen-2008 | Zanardi, F; Burreddu, P; Rassu, G; Auzzas, L; Battistini, L; Curti, C; Sartori, A; Nicastro, G; Menchi, G; Cini, N; Bottoncetti, A; Raspanti, S; Casiraghi, G | |
| The Practice of Ring Constraint in Peptidomimetics Using Bicyclic and Polycyclic Amino Acids. | 1-gen-2008 | Hanessian, S; Auzzas, L | |
| omega-Alkoxy analogues of SAHA(vorinostat) as inhibitors of HDAC: a study of chain-lenght and stereochemical dependence. | 1-gen-2007 | Hanessian S.; Auzzas L.; Giannini G.; Marzi M.; Cabri W.; Barbarino M.; Vesci L.; Pisano C. | |
| Exploring Alternative Zn-binding Groups in the Design of HDAC inhibitors: Squaric Acid, N-Hydroxyurea, and Oxazoline Analogues of SAHA | 1-gen-2006 | Hanessian S.; Vinci V.; Auzzas L.; Marzi M.; Giannini G. | |
| New Enantioselective Entry to Cycloheptane Amino Acid Polyols. | 1-gen-2006 | Curti C.; Zanardi F.; Battistini L.; Sartori A.; Rassu G.; Auzzas L.; Roggio A.; Pinna L.; Casiraghi G. | |
| Grafting Aminocyclopentane Carboxylic Acids onto the RGD Tripeptide Sequence Generates Low Nanomolar aVb3/aVb5 Integrin Dual Binders. | 1-gen-2005 | Casiraghi, G; Rassu, G; Auzzas, L; Burreddu, P; Gaetani, E; Battistini, L; Zanardi, F; Curti, C; Nicastro, G; Belvisi, L; Motto, I; Castorina, M; Giannini, G; Pisano, C | |
| Advances in the Chemical Synthesis of Medium-sized Cyclitols | 1-gen-2004 | Rassu, G; Auzzas, L; Battistini, L; Casiraghi, ; G, | |
| Enantioselective Total Synthesis of (1R,3S,4R,5R)-1-Amino-4,5-dihydroxycyclopentane-1,3-dicarboxylic Acid. A Full-Aldol Access to Carbaketose Derivatives | 1-gen-2004 | Battistini, L; Curti, C; Zanardi, F; Rassu, G; Auzzas, L; Casiraghi, G | |
| Variable Strategy toward Carbasugars and Relatives. 6. Diastereoselective Synthesis of 2-Deoxy-2-amino-5a-carba-beta-L-mannopyranuronic Acid and 2-Deoxy-2-amino-5a-carba-beta-L-mannopyranose | 1-gen-2004 | Rassu G.; Auzzas L.; Zambrano V.; Burreddu P.; Pinna L.; Battistini L.; Zanardi F.; Casiraghi G. | |
| A Short Entry to Novel (2)-Methyl Branched 4a-Carbafuranoses | 1-gen-2003 | Rassu, G; Auzzas, L; Zambrano, V; Burreddu, P; Battistini, L; Curti, C | |
| A short entry to novel C(2)-methyl branched 4a-carbafuranoses | 1-gen-2003 | Rassu, Gloria; Auzzas, Luciana; Zambrano, Vincenzo; Burreddu, Paola; Battistini, Lucia; Curti, Claudio | |
| Advances in Chemical Synthesis of Carbasugars and Analogues | 1-gen-2003 | Rassu, G; Auzzas, L; Pinna, L; Battistini, L; Curti, C | |
| Isopavines as a New Class of Morphinomimetics | 1-gen-2003 | Casiraghi, G; Zanardi, F; Auzzas, L; Appendino, G | |
| Variable Strategy toward Carbasugars and Relatives. 5. Focus on Preparation of Chiral Nonracemic Medium-Sized Carbocycles | 1-gen-2003 | Rassu, Gloria; Auzzas, Luciana; Pinna, Luigi; Zambrano, Vincenzo; Zanardi, Franca; Battistini, Lucia; Gaetani, Enrico; Curti, Claudio; Casiraghi, Giovanni | |
| Variable Strategy towards Carbasugars and Relatives. 5. Focus on Preparation of Chiral Nonracemic Medium-Sized Carbocycles | 1-gen-2003 | Rassu, G; Auzzas, L; Pinna, L; Zambrano, V; Zanardi, F; Battistini, L; Gaetani, E; Curti, C; Casiraghi, G |