DE SIMONE, GIUSEPPINA
DE SIMONE, GIUSEPPINA
Istituto di Biostrutture e Bioimmagini - IBB - Sede Napoli
Depsides from Origanum dictamnus and Satureja pilosa as selective inhibitors of carbonic anhydrases: Isolation, structure elucidation, X‐ray crystallography
2025 Paloukopoulou, Charikleia; Ntagli, Ogouschan Salim; Gherardi, Luca; Dourdouni, Virginia; Filippou, Glykeria; Alterio, Vincenzo; Giovannuzzi, Simone; Massardi, Maria Luisa; De Simone, Giuseppina; Ronca, Roberto; Supuran, Claudiu T.; Pescitelli, Gennaro; Karioti, Anastasia
Editorial: Emerging advancements in the carbonic anhydrase field
2025 Monti, Simona Maria; Alterio, Vincenzo; Parkkila, Seppo; Supuran, Claudiu T.; De Simone, Giuseppina
Fungal α-carbonic anhydrases
2025 D'Ambrosio, Katia; Di Fiore, Anna; Alterio, Vincenzo; Buonanno, Martina; Vivenzio, Vincenzo Massimiliano; Monti, Simona Maria; De Simone, Giuseppina; Langella, Emma
Multi-faceted exploration of the novel active γ-carbonic anhydrase PaCAγ1 in the human pathogen Pseudomonas aeruginosa
2025 Vivenzio, Vincenzo Massimiliano; Braga, Reygan; Bonardi, Alessandro; Alterio, Vincenzo; Scaloni, Andrea; Supuran, Claudiu T.; Patrauchan, Marianna A.; De Simone, Giuseppina; Monti, Simona Maria
Multiple Binding Modes of Inhibitors to Human Carbonic Anhydrases: An Update on the Design of Isoform-Specific Modulators of Activity
2025 D'Ambrosio, Katia; Di Fiore, Anna; Alterio, Vincenzo; Langella, Emma; Monti, Simona Maria; Supuran, Claudiu T.; De Simone, Giuseppina
Saccharomyces cerevesiae, Candida spp. and Cryptococcus neoformans β-CAs
2025 Di Fiore, Anna; Buonanno, Martina; Esposito, Davide; D'Ambrosio, Katia; Langella, Emma; De Simone, Giuseppina; Alterio, Vincenzo; Monti, Simona Maria
Anticancer drugs: where are we now?
2024 De Simone, Giuseppina; Supuran, Claudiu T.
Bacterial α-CAs: a biochemical and structural overview
2024 Vivenzio, Vincenzo Massimiliano; Esposito, Davide; Monti, Simona Maria; De Simone, Giuseppina
Exploring the binding mode of phenyl and vinyl boronic acids to human carbonic anhydrases
2024 Esposito, Davide; Monti, Simona Maria; Supuran, Claudiu T.; Winum, Jean-Yves; De Simone, Giuseppina; Alterio, Vincenzo
6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography
2023 Nocentini, Alessio; Bonardi, Alessandro; Bazzicalupi, Carla; Alterio, Vincenzo; Esposito, Davide; Monti, SIMONA MARIA; Smietana, Michael; DE SIMONE, Giuseppina; Supuran, Claudiu T.; Gratteri, Paola; Winum, Jean-Yves
A Combined in Silico and Structural Study Opens New Perspectives on Aliphatic Sulfonamides, a Still Poorly Investigated Class of CA Inhibitors
2023 Langella, Emma; Esposito, Davide; Monti, SIMONA MARIA; Supuran, Claudiu T.; DE SIMONE, Giuseppina; Alterio, Vincenzo
Carbonic anhydrase IX subcellular localization in normoxic and hypoxic SH-SY5Y neuroblastoma cells is assisted by its C-terminal protein interaction domain
2023 Succoio, Mariangela; Amiranda, Sara; Sasso, Emanuele; Marciano, Carmen; Finizio, Arianna; De Simone, Giuseppina; Garbi, Corrado; Zambrano, Nicola
Discovery of a novel series of potent carbonic anhydrase inhibitors with selective affinity for μ Opioid receptor for Safer and long-lasting analgesia
2023 Angeli, Andrea; Micheli, Laura; Turnaturi, Rita; Pasquinucci, Lorella; Parenti, Carmela; Alterio, Vincenzo; DI FIORE, Anna; DE SIMONE, Giuseppina; Monti, SIMONA MARIA; Carta, Fabrizio; Mannelli Lorenzo Di, Cesare; Ghelardini, Carla; Supuran Claudiu, T
Inhibition of Bone Marrow-Mesenchymal Stem Cell-Induced Carbonic Anhydrase IX Potentiates Chemotherapy Efficacy in Triple-Negative Breast Cancer Cells
2023 Sarnella, Annachiara; Ferrara, Ylenia; Albanese, Sandra; Omodei, Daniela; Cerchia, Laura; De Simone, Giuseppina; Supuran, Claudiu T; Zannetti, Antonella
Biochemical and Structural Insights into the Winged Helix Domain of P150, the Largest Subunit of the Chromatin Assembly Factor 1
2022 Ayoub, Joëlle; Buonanno, Martina; Di Fiore, Anna; De Simone, Giuseppina; Monti, Simona Maria
Biochemical, structural, and computational studies of a ?-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei
2022 Di Fiore, A; De Luca, V; Langella, E; Nocentini, A; Buonanno, M; Monti, Sm; Supuran, Ct; Capasso, C; De Simone, G
Inhibition of carbonic anhydrases IX/XII by SLC-0111 boosts cisplatin effects in hampering head and neck squamous carcinoma cell growth and invasion
2022 Sarnella, Annachiara; Ferrara, Ylenia; Auletta, Luigi; Albanese, Sandra; Cerchia, Laura; Alterio, Vincenzo; DE SIMONE, Giuseppina; Supuran, C. T.; Zannetti, Antonella
Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches
2022 Pagnozzi, Daniela; Pala, Nicolino; Biosa, Grazia; Dallocchio, Roberto; Dessì, Alessandro; Singh, Pankaj Kumar; Rogolino, Dominga; Di Fiore, Anna; De Simone, Giuseppina; Supuran, Claudiu T.; Sechi, Mario
Post-translational modifications in tumor-associated carbonic anhydrases
2022 DI FIORE, Anna; T Supuran, Claudiu; Scaloni, Andrea; DE SIMONE, Giuseppina
Sultam based Carbonic Anhydrase VII inhibitors for the management of neuropathic pain
2022 Akgül, Özlem; Lucarini, Elena; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; D'Ambrosio, Katia; Buonanno, Martina; Monti, Simona Maria; De Simone, Giuseppina; Angeli, Andrea; Supuran, Claudiu T.; Carta, Fabrizio
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Depsides from Origanum dictamnus and Satureja pilosa as selective inhibitors of carbonic anhydrases: Isolation, structure elucidation, X‐ray crystallography | 1-gen-2025 | Paloukopoulou, Charikleia; Ntagli, Ogouschan Salim; Gherardi, Luca; Dourdouni, Virginia; Filippou, Glykeria; Alterio, Vincenzo; Giovannuzzi, Simone; Massardi, Maria Luisa; De Simone, Giuseppina; Ronca, Roberto; Supuran, Claudiu T.; Pescitelli, Gennaro; Karioti, Anastasia | |
| Editorial: Emerging advancements in the carbonic anhydrase field | 1-gen-2025 | Monti, Simona Maria; Alterio, Vincenzo; Parkkila, Seppo; Supuran, Claudiu T.; De Simone, Giuseppina | |
| Fungal α-carbonic anhydrases | 1-gen-2025 | D'Ambrosio, Katia; Di Fiore, Anna; Alterio, Vincenzo; Buonanno, Martina; Vivenzio, Vincenzo Massimiliano; Monti, Simona Maria; De Simone, Giuseppina; Langella, Emma | |
| Multi-faceted exploration of the novel active γ-carbonic anhydrase PaCAγ1 in the human pathogen Pseudomonas aeruginosa | 1-gen-2025 | Vivenzio, Vincenzo Massimiliano; Braga, Reygan; Bonardi, Alessandro; Alterio, Vincenzo; Scaloni, Andrea; Supuran, Claudiu T.; Patrauchan, Marianna A.; De Simone, Giuseppina; Monti, Simona Maria | |
| Multiple Binding Modes of Inhibitors to Human Carbonic Anhydrases: An Update on the Design of Isoform-Specific Modulators of Activity | 1-gen-2025 | D'Ambrosio, Katia; Di Fiore, Anna; Alterio, Vincenzo; Langella, Emma; Monti, Simona Maria; Supuran, Claudiu T.; De Simone, Giuseppina | |
| Saccharomyces cerevesiae, Candida spp. and Cryptococcus neoformans β-CAs | 1-gen-2025 | Di Fiore, Anna; Buonanno, Martina; Esposito, Davide; D'Ambrosio, Katia; Langella, Emma; De Simone, Giuseppina; Alterio, Vincenzo; Monti, Simona Maria | |
| Anticancer drugs: where are we now? | 1-gen-2024 | De Simone, Giuseppina; Supuran, Claudiu T. | |
| Bacterial α-CAs: a biochemical and structural overview | 1-gen-2024 | Vivenzio, Vincenzo Massimiliano; Esposito, Davide; Monti, Simona Maria; De Simone, Giuseppina | |
| Exploring the binding mode of phenyl and vinyl boronic acids to human carbonic anhydrases | 1-gen-2024 | Esposito, Davide; Monti, Simona Maria; Supuran, Claudiu T.; Winum, Jean-Yves; De Simone, Giuseppina; Alterio, Vincenzo | |
| 6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography | 1-gen-2023 | Nocentini, Alessio; Bonardi, Alessandro; Bazzicalupi, Carla; Alterio, Vincenzo; Esposito, Davide; Monti, SIMONA MARIA; Smietana, Michael; DE SIMONE, Giuseppina; Supuran, Claudiu T.; Gratteri, Paola; Winum, Jean-Yves | |
| A Combined in Silico and Structural Study Opens New Perspectives on Aliphatic Sulfonamides, a Still Poorly Investigated Class of CA Inhibitors | 1-gen-2023 | Langella, Emma; Esposito, Davide; Monti, SIMONA MARIA; Supuran, Claudiu T.; DE SIMONE, Giuseppina; Alterio, Vincenzo | |
| Carbonic anhydrase IX subcellular localization in normoxic and hypoxic SH-SY5Y neuroblastoma cells is assisted by its C-terminal protein interaction domain | 1-gen-2023 | Succoio, Mariangela; Amiranda, Sara; Sasso, Emanuele; Marciano, Carmen; Finizio, Arianna; De Simone, Giuseppina; Garbi, Corrado; Zambrano, Nicola | |
| Discovery of a novel series of potent carbonic anhydrase inhibitors with selective affinity for μ Opioid receptor for Safer and long-lasting analgesia | 1-gen-2023 | Angeli, Andrea; Micheli, Laura; Turnaturi, Rita; Pasquinucci, Lorella; Parenti, Carmela; Alterio, Vincenzo; DI FIORE, Anna; DE SIMONE, Giuseppina; Monti, SIMONA MARIA; Carta, Fabrizio; Mannelli Lorenzo Di, Cesare; Ghelardini, Carla; Supuran Claudiu, T | |
| Inhibition of Bone Marrow-Mesenchymal Stem Cell-Induced Carbonic Anhydrase IX Potentiates Chemotherapy Efficacy in Triple-Negative Breast Cancer Cells | 1-gen-2023 | Sarnella, Annachiara; Ferrara, Ylenia; Albanese, Sandra; Omodei, Daniela; Cerchia, Laura; De Simone, Giuseppina; Supuran, Claudiu T; Zannetti, Antonella | |
| Biochemical and Structural Insights into the Winged Helix Domain of P150, the Largest Subunit of the Chromatin Assembly Factor 1 | 1-gen-2022 | Ayoub, Joëlle; Buonanno, Martina; Di Fiore, Anna; De Simone, Giuseppina; Monti, Simona Maria | |
| Biochemical, structural, and computational studies of a ?-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei | 1-gen-2022 | Di Fiore, A; De Luca, V; Langella, E; Nocentini, A; Buonanno, M; Monti, Sm; Supuran, Ct; Capasso, C; De Simone, G | |
| Inhibition of carbonic anhydrases IX/XII by SLC-0111 boosts cisplatin effects in hampering head and neck squamous carcinoma cell growth and invasion | 1-gen-2022 | Sarnella, Annachiara; Ferrara, Ylenia; Auletta, Luigi; Albanese, Sandra; Cerchia, Laura; Alterio, Vincenzo; DE SIMONE, Giuseppina; Supuran, C. T.; Zannetti, Antonella | |
| Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches | 1-gen-2022 | Pagnozzi, Daniela; Pala, Nicolino; Biosa, Grazia; Dallocchio, Roberto; Dessì, Alessandro; Singh, Pankaj Kumar; Rogolino, Dominga; Di Fiore, Anna; De Simone, Giuseppina; Supuran, Claudiu T.; Sechi, Mario | |
| Post-translational modifications in tumor-associated carbonic anhydrases | 1-gen-2022 | DI FIORE, Anna; T Supuran, Claudiu; Scaloni, Andrea; DE SIMONE, Giuseppina | |
| Sultam based Carbonic Anhydrase VII inhibitors for the management of neuropathic pain | 1-gen-2022 | Akgül, Özlem; Lucarini, Elena; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; D'Ambrosio, Katia; Buonanno, Martina; Monti, Simona Maria; De Simone, Giuseppina; Angeli, Andrea; Supuran, Claudiu T.; Carta, Fabrizio |