DE SIMONE, GIUSEPPINA

DE SIMONE, GIUSEPPINA  

Istituto di Biostrutture e Bioimmagini - IBB - Sede Napoli  

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Titolo Data di pubblicazione Autore(i) File
A Combined in Silico and Structural Study Opens New Perspectives on Aliphatic Sulfonamides, a Still Poorly Investigated Class of CA Inhibitors 1-gen-2023 Langella, Emma; Esposito, Davide; Monti, Simona Maria; Supuran, Claudiu T.; De Simone, Giuseppina; Alterio, Vincenzo
Biochemical, structural, and computational studies of a ?-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei 1-gen-2022 Di Fiore A.; De Luca V.; Langella E.; Nocentini A.; Buonanno M.; Monti S.M.; Supuran C.T.; Capasso C.; De Simone G.
Inhibition of carbonic anhydrases IX/XII by SLC-0111 boosts cisplatin effects in hampering head and neck squamous carcinoma cell growth and invasion 1-gen-2022 Sarnella, Annachiara; Ferrara, Ylenia; Auletta, Luigi; Albanese, Sandra; Cerchia, Laura; Alterio, Vincenzo; DE SIMONE, Giuseppina; Supuran, C. T.; Zannetti, Antonella
Post-translational modifications in tumor-associated carbonic anhydrases 1-gen-2022 DI FIORE, Anna; T Supuran, Claudiu; Scaloni, Andrea; DE SIMONE, Giuseppina
α-CAs from Photosynthetic Organisms 1-gen-2022 Langella, Emma; Di Fiore, Anna; Alterio, Vincenzo; Monti, Simona Maria; De Simone, Giuseppina; D’Ambrosio, Katia
Benzyl alcohol inhibits carbonic anhydrases by anchoring to the zinc coordinated water molecule 1-gen-2021 DE SIMONE, Giuseppina; Alterio, Vincenzo
The crystal structures of 2-(4-benzhydrylpiperazin-1-yl)-N-(4-sulfamoylphenyl)acetamide in complex with human carbonic anhydrase II and VII provide insights into selective CA inhibitor development 1-gen-2021 D'Ambrosio, Katia; DI FIORE, Anna; Buonanno, Martina; Kumari, Shikha; Tiwari, Manisha; Supuran Claudiu, T; Mishra Chandra, Bhushan; Monti, SIMONA MARIA; DE SIMONE, Giuseppina
Zeta-carbonic anhydrases show CS2 hydrolase activity: A new metabolic carbon acquisition pathway in diatoms? 1-gen-2021 Alterio, Vincenzo; Langella, Emma; Buonanno, Martina; Esposito, Davide; Nocentini, A.; Berrino, E.; Bua, S.; Polentarutti, M.; Supuran, C. T.; Monti, SIMONA MARIA; DE SIMONE, Giuseppina
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site 1-gen-2020 Bozdag, Murat; Supuran, Claudiu T.; Esposito, Davide; Angeli, Andrea; Carta, Fabrizio; Monti, Simona Maria; De Simone, Giuseppina; Alterio, Vincenzo
A Novel Inhibitor of Carbonic Anhydrases Prevents Hypoxia-Induced TNBC Cell Plasticity 1-gen-2020 Sarnella, Annachiara; D'Avino, Giuliana; Hill Billy, Samuel; Alterio, Vincenzo; Winum, Jeanyves; Supuran Claudiu, T; DE SIMONE, Giuseppina; Zannetti, Antonella
Biochemical and structural characterisation of a protozoan beta-carbonic anhydrase fromTrichomonas vaginalis 1-gen-2020 Urbanski, Linda J.; Di Fiore, Anna; Azizi, Latifeh; Hytonen, Vesa P.; Kuuslahti, Marianne; Buonanno, Martina; Monti, Simona M.; Angeli, Andrea; Emameh, Reza Zolfaghari; Supuran, Claudiu T.; De Simone, Giuseppina; Parkkila, Seppo
Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment 1-gen-2020 Angeli, Andrea; Carta, Fabrizio; Nocentini, Alessio; Winum, Jeanyves; Zalubovskis, Raivis; Akdemir, Atilla; Onnis, Valentina; Eldehna Wagdy, M; Capasso, Clemente; DE SIMONE, Giuseppina; Monti, SIMONA MARIA; Carradori, Simone; Donald William, A; Dedhar, Shoukat; Supuran Claudiu, T
Catechols: a new class of carbonic anhydrase inhibitors 1-gen-2020 D'Ambrosio, Katia; Carradori, Simone; Cesa, Stefania; Angeli, Andrea; Monti Simona, M; Supuran Claudiu, T; DE SIMONE, Giuseppina
Human Carbonic Anhydrases and Post-Translational Modifications: A Hidden World Possibly Affecting Protein Properties and Functions 1-gen-2020 DI FIORE, Anna; T Supuran, Claudiu; Scaloni, Andrea; DE SIMONE, Giuseppina
Inhibition of the newly discovered ?-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with inorganic anions and small molecules 1-gen-2020 Urbanski L.J.; Angeli A.; Hytonen V.P.; Di Fiore A.; Parkkila S.; De Simone G.; Supuran C.T.
Intrinsically disordered features of carbonic anhydrase IX proteoglycan-like domain 1-gen-2020 Langella, Emma; Buonanno, Martina; DE SIMONE, Giuseppina; Monti, SIMONA MARIA
Looking toward the Rim of the Active Site Cavity of Druggable Human Carbonic Anhydrase Isoforms 1-gen-2020 Mancuso, Francesca; Di Fiore, Anna; De Luca, Laura; Angeli, Andrea; Monti, Simona M.; De Simone, Giuseppina; Supuran, Claudiu T.; Gitto, Rosaria
Phenyl(thio)phosphon(amid)ate Benzenesulfonamides as Potent and Selective Inhibitors of Human Carbonic Anhydrases II and VII Counteract Allodynia in a Mouse Model of Oxaliplatin-Induced Neuropathy 1-gen-2020 Nocentini, Alessio; Alterio, Vincenzo; Bua, Silvia; Micheli, Laura; Esposito, Davide; Buonanno, Martina; Bartolucci, Gianluca; Osman, Sameh M.; ALOthman, Zeid A.; Cirilli, Roberto; Pierini, Marco; Monti, Simona Maria; Mannelli, Lorenzo Di Cesare; Gratteri, Paola; Ghelardini, Carla; De Simone, Giuseppina; Supuran, Claudiu T.
ALPHA-CARBONIC ANHYDRASES 1-gen-2019 DI FIORE, Anna; D'Ambrosio, Katia; Ayoub, Joelle; Alterio, Vincenzo; DE SIMONE, Giuseppina
Biochemical and Structural Insights into Carbonic Anhydrase XII/Fab6A10 Complex 1-gen-2019 Alterio, Vincenzo; Kellner, Markus; Esposito, Davide; Lieschestarnecker, Friederike; Bua, Silvia; Supuran Claudiu, T; Monti, SIMONA MARIA; Zeidler, Reinhard; DE SIMONE, Giuseppina