MAGA, GIOVANNI

MAGA, GIOVANNI  

Dipartimento di Scienze Biomediche - DSB  

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Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4- d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme 1-gen-2023 Poggialini F; Vagaggini C; Brai A; Pasqualini C; Crespan E; Maga G; Perini C; Cabella N; Botta L; Musumeci F; Frosini M; Schenone S; Dreassi E
Identification and Biological Characterization of the Pyrazolo[3,4-<i>d</i>]pyrimidine Derivative SI388 Active as Src Inhibitor 1-gen-2023 Contadini, C; Cirotti, C; Carbone, A; Norouzi, M; Cianciusi, A; Crespan, E; Perini, C; Maga, G; Barilà, D; Musumeci, F; Schenone, S
Interaction of SARS-CoV-2 Nucleocapsid Protein and Human RNA Helicases DDX1 and DDX3X Modulates Their Activities on Double-Stranded RNA 1-gen-2023 Lodola C; Secchi M; Sinigiani V; De Palma A; Rossi R; Perico D; Mauri PL; Maga G
DEAD-Box RNA Helicases DDX3X and DDX5 as Oncogenes or Oncosuppressors: A Network Perspective 1-gen-2022 Garbelli, A; Bione, S; Maga, G
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment 1-gen-2022 Di Maria, S; Picarazzi, F; Mori, M; Cianciusi, A; Carbone, A; Crespan, E; Perini, C; Sabetta, S; Deplano, S; Poggialini, F; Molinari, A; Aronne, R; Maccioni, E; Maga, G; Angelucci, A; Schenone, S; Musumeci, F; Dreassi, E
Privileged Scaffold Decoration for the Identification of the First Trisubstituted Triazine with Anti-SARS-CoV-2 Activity 1-gen-2022 Cesarini S; Vicenti I; Poggialini F; Secchi M; Giammarino F; Varasi I; Lodola C; Zazzi M; Dreassi E; Maga G; Botta L; Saladino R
Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors 1-gen-2022 Princiotto, S; Musso, L; Manetti, F; Marcellini, V; Maga, G; Crespan, E; Perini, C; Zaffaroni, N; Beretta, Gl; Dallavalle, S
A Role for Human DNA Polymerase lambda in Alternative Lengthening of Telomeres 1-gen-2021 Mentegari, E; Bertoletti, F; Kissova, M; Zucca, E; Galli, S; Tagliavini, G; Garbelli, A; Maffia, A; Bione, S; Ferrari, E; d'Adda di Fagagna, F; Francia, S; Sabbioneda, S; Chen, Ly; Lingner, J; Bergoglio, V; Hoffmann, Js; Hubscher, U; Crespan, E; Maga, G
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIII beta) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses 1-gen-2021 Grazia Martina M; Vicenti I; Bauer L; Crespan E; Rango E; Boccuto A; Olivieri N; Incerti M; Zwaagstra M; Allodi M; Bertoni S; Dreassi E; Zazzi M; van Kuppeveld FJM; Maga G; Radi M.
High flexibility of rnaseh2 catalytic activity with respect to non-canonical dna structures 1-gen-2021 Dede, M; Napolitano, S; Melati, A; Pirota, V; Maga, G; Crespan, E
System-oriented optimization of multi-target 2,6-diaminopurine derivatives: Easily accessible broad-spectrum antivirals active against flaviviruses, influenza virus and SARS-CoV-2 1-gen-2021 Vicenti, I; Martina, Mg; Boccuto, A; De Angelis, M; Giavarini, G; Dragoni, F; Marchi, S; Trombetta, Cm; Crespan, E; Maga, G; Eydoux, C; Decroly, E; Montomoli, E; Nencioni, L; Zazzi, M; Radi, M
Targeting ddx3x helicase activity with ba103 shows promising therapeutic effects in preclinical glioblastoma models 1-gen-2021 Brai A; Riva V; Clementi L; Falsitta L; Zamperini C; Sinigiani V; Festuccia C; Sabetta S; Aiello D; Roselli C; Garbelli A; Trivisani CI; Maccari L; Bugli F; Sanguinetti M; Calandro P; Chiariello M; Quaranta P; Botta L; Angelucci A; Maga G; Botta M.
A Structural View of SARS-CoV-2 RNA Replication Machinery: RNA Synthesis, Proofreading and Final Capping 1-gen-2020 Romano, M; Ruggiero, A; Squeglia, F; Maga, G; Berisio, R
DDX3X Inhibitors, an Effective Way to Overcome HIV-1 Resistance Targeting Host Proteins 1-gen-2020 Brai A; Riva V; Saladini F; Zamperini C; Trivisani CI; Garbelli A; Pennisi C; Giannini A; Boccuto A; Bugli F; Martini M; Sanguinetti M; Zazzi M; Dreassi E; Botta M; Maga G.
Exploring the Implication of DDX3X in DENV Infection: Discovery of the First-in-Class DDX3X Fluorescent Inhibitor 1-gen-2020 Brai, A; Boccuto, A; Monti, M; Marchi, S; Vicenti, I; Saladini, F; Trivisani, Ci; Pollutri, A; Trombetta, Cm; Montomoli, E; Riva, V; Garbelli, A; Nola, Em; Zazzi, M; Maga, G; Dreassi, E; Botta, M
Host DDX Helicases as Possible SARS-CoV-2 Proviral Factors: A Structural Overview of Their Hijacking Through Multiple Viral Proteins 1-gen-2020 Squeglia, F; Romano, M; Ruggiero, A; Maga, G; Berisio, R
New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains 1-gen-2020 Nalli, M; Armijos Rivera, Ji; Masci, D; Coluccia, A; Badia, R; Riveiramuñoz, E; Brambilla, A; Cinquina, E; Turriziani, O; Falasca, F; Catalano, M; Limatola, C; Esté, Ja; Maga, G; Silvestri, R; Crespan, E; La Regina, G
Novel alternative ribonucleotide excision repair pathways in human cells by DDX3X and specialized DNA polymerases 1-gen-2020 Riva V; Garbelli A; Casiraghi F; Arena F; Trivisani CI; Gagliardi A; Bini L; Schroeder M; Maffia A; Sabbioneda S; Maga G.
Novel Insights into the Biochemical Mechanism of CK1epsilon and its Functional Interplay with DDX3X 1-gen-2020 Bono, B; Franco, G; Riva, V; Garbelli, A; Maga, G
Plant Molecular Farming as a Strategy Against COVID-19 - The Italian Perspective 1-gen-2020 Lico C.; Santi L.; Baschieri S.; Noris E.; Marusic C.; Donini M.; Pedrazzini E.; Maga G.; Franconi R.; Di Bonito P.; Avesani L.