GIORDANO, ASSUNTA
GIORDANO, ASSUNTA
Istituto di Chimica Biomolecolare - ICB - Sede Pozzuoli
Identification and development of BRD9 chemical probes
2024 Colarusso, Ester; Giovanna Chini, Maria; Bifulco, Giuseppe; Lauro, Gianluigi; Giordano, Assunta
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole‐Based Inhibitors of Soluble Epoxide Hydrolase (sEH)
2024 Gazzillo, Erica; Colarusso, Ester; Giordano, Assunta; Chini, Maria Giovanna; Potenza, Marianna; Hofstetter, Robert Klaus; Iorizzi, Maria; Werz, Oliver; Lauro, Gianluigi; Bifulco, Giuseppe
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders
2023 Colarusso, Ester; Ceccacci, Sara; Chiara Monti, Maria; Gazzillo, Erica; Giordano, Assunta; Giovanna Chini, Maria; Grazia Ferraro, Maria; Piccolo, Marialuisa; Irace, Carlo; Bifulco, Giuseppe; Lauro, Gianluigi
Identification of 2-aminoacyl-1,3,4-thiadiazoles as prostaglandin E2 and leukotriene biosynthesis inhibitors
2023 Potenza, Marianna; Giordano, Assunta; G Chini, Maria; Saviano, Anella; Kretzer, Christian; Raucci, Federica; Russo, Marina; Lauro, Gianluigi; Terracciano, Stefania; Bruno, Ines; Iorizzi, Maria; K Hofstetter, Robert; Pace, Simona; Maione, Francesco; Werz, Oliver; Bifulco, Giuseppe
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis
2022 Colarusso, Ester; Gazzillo, Erica; Boccia, Eleonora; Giordano, Assunta; Giovanna Chini, Maria; Bifulco, Giuseppe; Lauro, Gianluigi
Repositioning of quinazolinedione-based compounds on soluble epoxide hydrolase (sEH) through 3D structure-based pharmacophore model-driven investigation.
2022 Gazzillo, E; Terracciano, S; Ruggiero, D; Potenza, M; Chini, Mg; Lauro, G; Fischer, K; Hofstetter, Rk; Giordano, A; Werz, O; Bruno, I; Bifulco, G
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways
2021 Potenza, Marianna; Sciarretta, Martina; Giovanna Chini, Maria; Saviano, Anella; Maione, Francesco; Valeria D'Auria, Maria; De Marino, Simona; Giordano, Assunta; Klaus Hofstetter, Robert; Festa, Carmen; Werz, Oliver; Bifulco, Giuseppe
Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE(2) Levels
2020 Chini Maria, G; Giordano, Assunta; Potenza, Marianna; Terracciano, Stefania; Fischer, Katrin; Vaccaro Maria, C; Colarusso, Ester; Bruno, Ines; Riccio, Raffaele; Koeberle, Andreas; Werz, Oliver; Bifulco, Giuseppe
Identification of the 2-benzoxazol-2-yl-phenol scaffold as new hit for JMJD3 inhibition
2019 Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; C Scala, Maria; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone
Discovery of new erbB4 inhibitors: Repositioning an orphan chemical library by inverse virtual screening
2018 Assunta Giordano; Giovanni Forte; Luigia Massimo; Raffaele Riccio; Giuseppe Bifulco; Raffaele Riccio; Simone Di Micco
Virtual fragment screening identification of a novel Quinoline-5,8- dicarboxylic acid derivative as selective JMJD3 inhibitor
2018 Giordano, Assunta; Del Gaudio, Federica; Johansson, Catrine; Riccio, Raffaele; Oppermann, Udo; Di Micco, Simone
Combinatorial approach for the discovery of novel microsomal prostaglandin E 2 synthase - 1 (mPGES - 1) inhibitors
2017 Giovanna Chini, Maria; Giordano, Assunta; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Riccio, Raffaele; Cantone, Vincenza; Werz, Oliver; Bifulco, Giuseppe
Identification of new Erb B 4 inhibitors by inverse virtual screening
2017 Giordano, Assunta; Forte, Giovanni; Dal Piaz, Fabrizio; del Gaudio, Federica; De Tommasi, Nunziatina; Gazzerro, Patrizia; Riccio, Raffaele; Bifulco, Giuseppe; Di Micco, Simone
Aureivirga marina gen. nov., sp. nov., a novel marine bacterium isolated from the Mediterranean sponge Axinella verrucosa
2013 Haber, M; Shefer, S; Giordano, A; Orlando, P; Gambacorta, A; Ilan, M
Biochemical phenotype of a common disease-causing mutation and a possible therapeutic approach for the phosphomannomutase 2-associated disorder of glycosylation
2013 Andreotti, Giuseppina; Pedone, Emilia; Giordano, Assunta; Vittoria Cubellis, Maria
Fulvitalea axinellae gen. nov., sp. nov., a novel member of the family Flammeovirgaceae isolated from the Mediterranean sponge Axinella verrucosa
2013 Haber, M; Shefer, S; Giordano, A; Orlando, P; Gambacorta, A; Ilan, M
Luteivirga sdotyamensis gen. nov., sp. nov., a novel bacterium of the phylum Bacteroidetes isolated from the Mediterranean sponge Axinella polypoides
2013 Haber, M; Shefer, S; Giordano, A; Orlando, P; Gambacorta, A; Ilan, M
New bacteroidetes bacteria associated with mediterranean Axinella sponges
2012 Haber M; Shefer S; Giordano A; Orlando P; Gambacorta A; Illan; M
Pseudomonas litolaris sp. nov., isolated from mediterranean seawater
2012 Pascual, J; Lucena, T; Ruvira, ; Ma, ; Giordano, A; Gambacorta, A; Garay, E; Arahal, ; D, R; Pujalte, ; M, J; Macian, ; C,
Pseudomonas litoralis sp. nov., isolated from Mediterranean seawater
2012 Pascual J; Lucena T; Ruvira MA; Giordano A; Gambacorta A; Garay E; Arahal DR; Pujalte MJ; Macian MC
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Identification and development of BRD9 chemical probes | 1-gen-2024 | Colarusso, Ester; Giovanna Chini, Maria; Bifulco, Giuseppe; Lauro, Gianluigi; Giordano, Assunta | |
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole‐Based Inhibitors of Soluble Epoxide Hydrolase (sEH) | 1-gen-2024 | Gazzillo, Erica; Colarusso, Ester; Giordano, Assunta; Chini, Maria Giovanna; Potenza, Marianna; Hofstetter, Robert Klaus; Iorizzi, Maria; Werz, Oliver; Lauro, Gianluigi; Bifulco, Giuseppe | |
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders | 1-gen-2023 | Colarusso, Ester; Ceccacci, Sara; Chiara Monti, Maria; Gazzillo, Erica; Giordano, Assunta; Giovanna Chini, Maria; Grazia Ferraro, Maria; Piccolo, Marialuisa; Irace, Carlo; Bifulco, Giuseppe; Lauro, Gianluigi | |
Identification of 2-aminoacyl-1,3,4-thiadiazoles as prostaglandin E2 and leukotriene biosynthesis inhibitors | 1-gen-2023 | Potenza, Marianna; Giordano, Assunta; G Chini, Maria; Saviano, Anella; Kretzer, Christian; Raucci, Federica; Russo, Marina; Lauro, Gianluigi; Terracciano, Stefania; Bruno, Ines; Iorizzi, Maria; K Hofstetter, Robert; Pace, Simona; Maione, Francesco; Werz, Oliver; Bifulco, Giuseppe | |
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis | 1-gen-2022 | Colarusso, Ester; Gazzillo, Erica; Boccia, Eleonora; Giordano, Assunta; Giovanna Chini, Maria; Bifulco, Giuseppe; Lauro, Gianluigi | |
Repositioning of quinazolinedione-based compounds on soluble epoxide hydrolase (sEH) through 3D structure-based pharmacophore model-driven investigation. | 1-gen-2022 | Gazzillo, E; Terracciano, S; Ruggiero, D; Potenza, M; Chini, Mg; Lauro, G; Fischer, K; Hofstetter, Rk; Giordano, A; Werz, O; Bruno, I; Bifulco, G | |
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways | 1-gen-2021 | Potenza, Marianna; Sciarretta, Martina; Giovanna Chini, Maria; Saviano, Anella; Maione, Francesco; Valeria D'Auria, Maria; De Marino, Simona; Giordano, Assunta; Klaus Hofstetter, Robert; Festa, Carmen; Werz, Oliver; Bifulco, Giuseppe | |
Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE(2) Levels | 1-gen-2020 | Chini Maria, G; Giordano, Assunta; Potenza, Marianna; Terracciano, Stefania; Fischer, Katrin; Vaccaro Maria, C; Colarusso, Ester; Bruno, Ines; Riccio, Raffaele; Koeberle, Andreas; Werz, Oliver; Bifulco, Giuseppe | |
Identification of the 2-benzoxazol-2-yl-phenol scaffold as new hit for JMJD3 inhibition | 1-gen-2019 | Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; C Scala, Maria; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone | |
Discovery of new erbB4 inhibitors: Repositioning an orphan chemical library by inverse virtual screening | 1-gen-2018 | Assunta Giordano; Giovanni Forte; Luigia Massimo; Raffaele Riccio; Giuseppe Bifulco; Raffaele Riccio; Simone Di Micco | |
Virtual fragment screening identification of a novel Quinoline-5,8- dicarboxylic acid derivative as selective JMJD3 inhibitor | 1-gen-2018 | Giordano, Assunta; Del Gaudio, Federica; Johansson, Catrine; Riccio, Raffaele; Oppermann, Udo; Di Micco, Simone | |
Combinatorial approach for the discovery of novel microsomal prostaglandin E 2 synthase - 1 (mPGES - 1) inhibitors | 1-gen-2017 | Giovanna Chini, Maria; Giordano, Assunta; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Riccio, Raffaele; Cantone, Vincenza; Werz, Oliver; Bifulco, Giuseppe | |
Identification of new Erb B 4 inhibitors by inverse virtual screening | 1-gen-2017 | Giordano, Assunta; Forte, Giovanni; Dal Piaz, Fabrizio; del Gaudio, Federica; De Tommasi, Nunziatina; Gazzerro, Patrizia; Riccio, Raffaele; Bifulco, Giuseppe; Di Micco, Simone | |
Aureivirga marina gen. nov., sp. nov., a novel marine bacterium isolated from the Mediterranean sponge Axinella verrucosa | 1-gen-2013 | Haber, M; Shefer, S; Giordano, A; Orlando, P; Gambacorta, A; Ilan, M | |
Biochemical phenotype of a common disease-causing mutation and a possible therapeutic approach for the phosphomannomutase 2-associated disorder of glycosylation | 1-gen-2013 | Andreotti, Giuseppina; Pedone, Emilia; Giordano, Assunta; Vittoria Cubellis, Maria | |
Fulvitalea axinellae gen. nov., sp. nov., a novel member of the family Flammeovirgaceae isolated from the Mediterranean sponge Axinella verrucosa | 1-gen-2013 | Haber, M; Shefer, S; Giordano, A; Orlando, P; Gambacorta, A; Ilan, M | |
Luteivirga sdotyamensis gen. nov., sp. nov., a novel bacterium of the phylum Bacteroidetes isolated from the Mediterranean sponge Axinella polypoides | 1-gen-2013 | Haber, M; Shefer, S; Giordano, A; Orlando, P; Gambacorta, A; Ilan, M | |
New bacteroidetes bacteria associated with mediterranean Axinella sponges | 1-gen-2012 | Haber M; Shefer S; Giordano A; Orlando P; Gambacorta A; Illan; M | |
Pseudomonas litolaris sp. nov., isolated from mediterranean seawater | 1-gen-2012 | Pascual, J; Lucena, T; Ruvira, ; Ma, ; Giordano, A; Gambacorta, A; Garay, E; Arahal, ; D, R; Pujalte, ; M, J; Macian, ; C, | |
Pseudomonas litoralis sp. nov., isolated from Mediterranean seawater | 1-gen-2012 | Pascual J; Lucena T; Ruvira MA; Giordano A; Gambacorta A; Garay E; Arahal DR; Pujalte MJ; Macian MC |