AROSIO, DANIELA
AROSIO, DANIELA
Istituto di Scienze e Tecnologie Chimiche "Giulio Natta" - SCITEC - Sede Secondaria Milano - Via C. Golgi
A combined approach of structure-based virtual screening and NMR to interrupt the PD-1/PD-L1 axis: Biphenyl-benzimidazole containing compounds as novel PD-L1 inhibitors
2024 Donati, Greta; Viviano, Monica; D'Amore Vincenzo, M.; Cipriano, Alessandra; Diakogiannaki, Isidora; Amato, Jussara; Tomassi, Stefano; Brancaccio, Diego; Russomanno, Pasquale; Di Leva Francesco, S.; Arosio, Daniela; Seneci, Pierfausto; Taliani, Sabrina; Magiera-Mularz, Katarzyna; Musielak, Bogdan; Skalniak, Lukasz; Holak Tad, A.; Castellano, Sabrina; La Pietra, Valeria; Marinelli, Luciana
Novel, soluble 3-heteroaryl-substituted tanshinone mimics attenuate the inflammatory response in murine macrophages
2024 Facen, Elisa.; Assoni, Giulia.; Donati, Greta.; Paladino, Dalila.; Carreira, Agata.; Bonomo, Isabel.; La Pietra, Valeria; Lotti, Roberta; Houser, Josef; Fava Luca, L.; Seneci, Pierfausto.; Marinelli, Luciana; Arosio, Daniela; Provenzani, Alessandro
HuR modulation counteracts lipopolysaccharide response in murine macrophages
2023 Bonomo, I; Assoni, G; La Pietra, V; Canarutto, G; Facen, E; Donati, G; Zucal, C; Genovese, S; Micaelli, M; Perezrafols, A; Robbiati, S; Kontoyannis, Dl; De Matteo, M; Fragai, M; Seneci, P; Marinelli, L; Arosio, D; Piazza, S; Provenzani, A
RGD Cyclopeptide Equipped with a Lysine-Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency
2023 Sacco, Giovanni; Arosio, Daniela; Paolillo, Mayra; Gloger, Andreas; Scheuermann, Jorg; Pignataro, Luca; Belvisi, Laura; Dal Corso, Alberto; Gennari, Cesare
Theoretical and experimental studies on the interaction of biphenyl ligands with human and murine PD-L1: Up-to-date clues for drug design
2023 Donati, Greta; D'Amore Vincenzo, Maria; Russomanno, Pasquale; Cerofolini, Linda; Amato, Jussara; Marzano, Simona; Salobehaj, Maria; Rizzo, Domenico; Assoni, Giulia; Carotenuto, Alfonso; La Pietra, Valeria; Arosio, Daniela; Seneci, Pierfausto; Fragai, Marco; Brancaccio, Diego; Di Leva Francesco, Saverio; Marinelli, Luciana
HuR-targeted agents: An insight into medicinal chemistry, biophysical, computational studies and pharmacological effects on cancer models
2022 Assoni, Giulia; La Pietra, Valeria; Digilio, Rosangela; Ciani, Caterina; Licata Nausicaa, Valentina; Micaelli, Mariachiara; Facen, Elisa; Tomaszewska, Weronika; Cerofolini, Linda; Pérezràfols, Anna; Varela Rey, Marta; Fragai, Marco; Woodhoo, Ashwin; Marinelli, Luciana; Arosio, Daniela; Bonomo, Isabelle; Provenzani, Alessandro; Seneci, Pierfausto
Squalene-Based Nano-Assemblies Improve the Pro-Autophagic Activity of Trehalose
2022 Frapporti, Giulia; Colombo, Eleonora; Ahmed, Hazem; Assoni, Giulia; Polito, Laura; Randazzo, Pietro; Arosio, Daniela; Seneci, Pierfausto; Piccoli, Giovanni
Interfering with the Tumor-Immune Interface: Making Way for Triazine-Based Small Molecules as Novel PD-L1 Inhibitors
2021 Russomanno, Pasquale; Assoni, Giulia; Amato, Jussara; D'Amore, Vincenzo Maria; Scaglia, Riccardo; Brancaccio, Diego; Pedrini, Martina; Polcaro, Giovanna; La Pietra, Valeria; Orlando, Paolo; Falzoni, Marianna; Cerofolini, Linda; Giuntini, Stefano; Fragai, Marco; Pagano, Bruno; Donati, Greta; Novellino, Ettore; Quintavalle, Cristina; Condorelli, Gerolama; Sabbatino, Francesco; Seneci, Pierfausto; Arosio, Daniela; Pepe, Stefano; Marinelli, Luciana
Trehalose-based neuroprotective autophagy inducers
2021 Assoni, Giulia; Frapporti, Giulia; Colombo, Eleonora; Gornati, Davide; PerezCarrion Maria, Dolores; Polito, Laura; Seneci, Pierfausto; Piccoli, Giovanni; Arosio, Daniela
Cyclic RGD and iso DGR Integrin Ligands Containing cis-2-amino-1-cyclopentanecarboxylic ( cis-Beta-ACPC) Scaffolds
2020 Panzeri, Silvia; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Civera, Monica; Potenza, Donatella; Vasile, Francesca; Kemker, Isabell; Ertl, Thomas; Sewald, Norbert; Reiser, Oliver; Piarulli, Umberto
Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake
2020 Pina, Arianna; Kadri, Malika; Arosio, Daniela; Dal Corso, Alberto; Coll, Jeanluc; Gennari, Cesare; Boturyn, Didier
Shifting Towards alpha(V)beta(6)Integrin Ligands Using Novel Aminoproline-Based Cyclic Peptidomimetics
2020 Bugatti, Kelly; Bruno, Agostino; Arosio, Daniela; Sartori, Andrea; Curti, Claudio; Augustijn, Lisa; Zanardi, Franca; Battistini, Lucia
A dimeric bicyclic RGD ligand displays enhanced integrin binding affinity and strong biological effects on U-373 MG glioblastoma cells
2019 Sacco, Giovanni; Dal Corso, Alberto; Arosio, Daniela; Belvisi, Laura; Paolillo, Mayra; Pignataro, Luca; Gennari, Cesare
beta-Glucuronidase triggers extracellular MMAE release from an integrin-targeted conjugate
2019 Rivas, Paula Lopez; Mueller, Christoph; Breunig, Christian; Hechler, Torsten; Pahl, Andreas; Arosio, Daniela; Belvisi, Laura; Pignataro, Luca; Dal Corso, Alberto; Gennari, Cesare
Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery
2019 Borbély, Adina; Figueras, Eduard; Martins, Ana; Bodero, Lizeth; Raposo Moreira Dias, André; López Rivas, Paula; Pina, Arianna; Arosio, Daniela; Gallinari, Paola; Frese, Marcel; Steinkühler, Christian; Gennari, Cesare; Piarulli, Umberto; Sewald, Norbert
Intracisternal delivery of PEG-coated gold nanoparticles results in high brain penetrance and long-lasting stability
2019 Spinelli, Antonello; Girelli, Maria; Arosio, Daniela; Polito, Laura; Podini, Paola; Martino, Gianvito; Seneci, Pierfausto; Muzio, Luca; Menegon, Andrea
Kiss and Run: Promoting Effective and Targeted Cellular Uptake of a Drug Delivery Vehicle Composed of an Integrin-Targeting Diketopiperazine Peptidomimetic and a Cell-Penetrating Peptide
2019 Feni, Lucia; Parente, Sara; Robert, Clémence; Gazzola, Silvia; Arosio, Daniela; Piarulli, Umberto; Neundorf, Ines
Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate
2019 Andre Raposo Moreira Dias; Arianna Pina; Amelia Dean; HansGeorg Lerchen; Michele Caruso;Fabio Gasparri; Ivan Fraietta; Sonia Troiani; Daniela Arosio; Laura Belvisi; Luca Pignataro; Alberto Dal Corso; Cesare Gennari
Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors
2019 Zanella, Simone; Bocchinfuso, Gianfranco; De Zotti, Marta; Arosio, Daniela; Marino, Franca; Raniolo, Stefano; Pignataro, Luca; Sacco, Giovanni; Palleschi, Antonio; Siano Alvaro, S; Piarulli, Umberto; Belvisi, Laura; Formaggio, Fernando; Gennari, Cesare; Stella, Lorenzo
Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin (V3)
2019 Dias Andre Raposo, Moreira; Bodero, Lizeth; Martins, Ana; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Pignataro, Luca; Steinkuhler, Christian; Dal Corso, Alberto; Gennari, Cesare; Piarulli, Umberto
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A combined approach of structure-based virtual screening and NMR to interrupt the PD-1/PD-L1 axis: Biphenyl-benzimidazole containing compounds as novel PD-L1 inhibitors | 1-gen-2024 | Donati, Greta; Viviano, Monica; D'Amore Vincenzo, M.; Cipriano, Alessandra; Diakogiannaki, Isidora; Amato, Jussara; Tomassi, Stefano; Brancaccio, Diego; Russomanno, Pasquale; Di Leva Francesco, S.; Arosio, Daniela; Seneci, Pierfausto; Taliani, Sabrina; Magiera-Mularz, Katarzyna; Musielak, Bogdan; Skalniak, Lukasz; Holak Tad, A.; Castellano, Sabrina; La Pietra, Valeria; Marinelli, Luciana | |
| Novel, soluble 3-heteroaryl-substituted tanshinone mimics attenuate the inflammatory response in murine macrophages | 1-gen-2024 | Facen, Elisa.; Assoni, Giulia.; Donati, Greta.; Paladino, Dalila.; Carreira, Agata.; Bonomo, Isabel.; La Pietra, Valeria; Lotti, Roberta; Houser, Josef; Fava Luca, L.; Seneci, Pierfausto.; Marinelli, Luciana; Arosio, Daniela; Provenzani, Alessandro | |
| HuR modulation counteracts lipopolysaccharide response in murine macrophages | 1-gen-2023 | Bonomo, I; Assoni, G; La Pietra, V; Canarutto, G; Facen, E; Donati, G; Zucal, C; Genovese, S; Micaelli, M; Perezrafols, A; Robbiati, S; Kontoyannis, Dl; De Matteo, M; Fragai, M; Seneci, P; Marinelli, L; Arosio, D; Piazza, S; Provenzani, A | |
| RGD Cyclopeptide Equipped with a Lysine-Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency | 1-gen-2023 | Sacco, Giovanni; Arosio, Daniela; Paolillo, Mayra; Gloger, Andreas; Scheuermann, Jorg; Pignataro, Luca; Belvisi, Laura; Dal Corso, Alberto; Gennari, Cesare | |
| Theoretical and experimental studies on the interaction of biphenyl ligands with human and murine PD-L1: Up-to-date clues for drug design | 1-gen-2023 | Donati, Greta; D'Amore Vincenzo, Maria; Russomanno, Pasquale; Cerofolini, Linda; Amato, Jussara; Marzano, Simona; Salobehaj, Maria; Rizzo, Domenico; Assoni, Giulia; Carotenuto, Alfonso; La Pietra, Valeria; Arosio, Daniela; Seneci, Pierfausto; Fragai, Marco; Brancaccio, Diego; Di Leva Francesco, Saverio; Marinelli, Luciana | |
| HuR-targeted agents: An insight into medicinal chemistry, biophysical, computational studies and pharmacological effects on cancer models | 1-gen-2022 | Assoni, Giulia; La Pietra, Valeria; Digilio, Rosangela; Ciani, Caterina; Licata Nausicaa, Valentina; Micaelli, Mariachiara; Facen, Elisa; Tomaszewska, Weronika; Cerofolini, Linda; Pérezràfols, Anna; Varela Rey, Marta; Fragai, Marco; Woodhoo, Ashwin; Marinelli, Luciana; Arosio, Daniela; Bonomo, Isabelle; Provenzani, Alessandro; Seneci, Pierfausto | |
| Squalene-Based Nano-Assemblies Improve the Pro-Autophagic Activity of Trehalose | 1-gen-2022 | Frapporti, Giulia; Colombo, Eleonora; Ahmed, Hazem; Assoni, Giulia; Polito, Laura; Randazzo, Pietro; Arosio, Daniela; Seneci, Pierfausto; Piccoli, Giovanni | |
| Interfering with the Tumor-Immune Interface: Making Way for Triazine-Based Small Molecules as Novel PD-L1 Inhibitors | 1-gen-2021 | Russomanno, Pasquale; Assoni, Giulia; Amato, Jussara; D'Amore, Vincenzo Maria; Scaglia, Riccardo; Brancaccio, Diego; Pedrini, Martina; Polcaro, Giovanna; La Pietra, Valeria; Orlando, Paolo; Falzoni, Marianna; Cerofolini, Linda; Giuntini, Stefano; Fragai, Marco; Pagano, Bruno; Donati, Greta; Novellino, Ettore; Quintavalle, Cristina; Condorelli, Gerolama; Sabbatino, Francesco; Seneci, Pierfausto; Arosio, Daniela; Pepe, Stefano; Marinelli, Luciana | |
| Trehalose-based neuroprotective autophagy inducers | 1-gen-2021 | Assoni, Giulia; Frapporti, Giulia; Colombo, Eleonora; Gornati, Davide; PerezCarrion Maria, Dolores; Polito, Laura; Seneci, Pierfausto; Piccoli, Giovanni; Arosio, Daniela | |
| Cyclic RGD and iso DGR Integrin Ligands Containing cis-2-amino-1-cyclopentanecarboxylic ( cis-Beta-ACPC) Scaffolds | 1-gen-2020 | Panzeri, Silvia; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Civera, Monica; Potenza, Donatella; Vasile, Francesca; Kemker, Isabell; Ertl, Thomas; Sewald, Norbert; Reiser, Oliver; Piarulli, Umberto | |
| Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake | 1-gen-2020 | Pina, Arianna; Kadri, Malika; Arosio, Daniela; Dal Corso, Alberto; Coll, Jeanluc; Gennari, Cesare; Boturyn, Didier | |
| Shifting Towards alpha(V)beta(6)Integrin Ligands Using Novel Aminoproline-Based Cyclic Peptidomimetics | 1-gen-2020 | Bugatti, Kelly; Bruno, Agostino; Arosio, Daniela; Sartori, Andrea; Curti, Claudio; Augustijn, Lisa; Zanardi, Franca; Battistini, Lucia | |
| A dimeric bicyclic RGD ligand displays enhanced integrin binding affinity and strong biological effects on U-373 MG glioblastoma cells | 1-gen-2019 | Sacco, Giovanni; Dal Corso, Alberto; Arosio, Daniela; Belvisi, Laura; Paolillo, Mayra; Pignataro, Luca; Gennari, Cesare | |
| beta-Glucuronidase triggers extracellular MMAE release from an integrin-targeted conjugate | 1-gen-2019 | Rivas, Paula Lopez; Mueller, Christoph; Breunig, Christian; Hechler, Torsten; Pahl, Andreas; Arosio, Daniela; Belvisi, Laura; Pignataro, Luca; Dal Corso, Alberto; Gennari, Cesare | |
| Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery | 1-gen-2019 | Borbély, Adina; Figueras, Eduard; Martins, Ana; Bodero, Lizeth; Raposo Moreira Dias, André; López Rivas, Paula; Pina, Arianna; Arosio, Daniela; Gallinari, Paola; Frese, Marcel; Steinkühler, Christian; Gennari, Cesare; Piarulli, Umberto; Sewald, Norbert | |
| Intracisternal delivery of PEG-coated gold nanoparticles results in high brain penetrance and long-lasting stability | 1-gen-2019 | Spinelli, Antonello; Girelli, Maria; Arosio, Daniela; Polito, Laura; Podini, Paola; Martino, Gianvito; Seneci, Pierfausto; Muzio, Luca; Menegon, Andrea | |
| Kiss and Run: Promoting Effective and Targeted Cellular Uptake of a Drug Delivery Vehicle Composed of an Integrin-Targeting Diketopiperazine Peptidomimetic and a Cell-Penetrating Peptide | 1-gen-2019 | Feni, Lucia; Parente, Sara; Robert, Clémence; Gazzola, Silvia; Arosio, Daniela; Piarulli, Umberto; Neundorf, Ines | |
| Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate | 1-gen-2019 | Andre Raposo Moreira Dias; Arianna Pina; Amelia Dean; HansGeorg Lerchen; Michele Caruso;Fabio Gasparri; Ivan Fraietta; Sonia Troiani; Daniela Arosio; Laura Belvisi; Luca Pignataro; Alberto Dal Corso; Cesare Gennari | |
| Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors | 1-gen-2019 | Zanella, Simone; Bocchinfuso, Gianfranco; De Zotti, Marta; Arosio, Daniela; Marino, Franca; Raniolo, Stefano; Pignataro, Luca; Sacco, Giovanni; Palleschi, Antonio; Siano Alvaro, S; Piarulli, Umberto; Belvisi, Laura; Formaggio, Fernando; Gennari, Cesare; Stella, Lorenzo | |
| Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin (V3) | 1-gen-2019 | Dias Andre Raposo, Moreira; Bodero, Lizeth; Martins, Ana; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Pignataro, Luca; Steinkuhler, Christian; Dal Corso, Alberto; Gennari, Cesare; Piarulli, Umberto |